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(3S,4R)-1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-{[2-(1-ethylpiperidin-3-yl)-1H-imidazol-1-yl]methyl}-5-methylpyrazine
2-methyl-1-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-indole
(1S,5R)-6-(4-methylpyridine-3-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
3-[4-(3-methylpyridin-4-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
2-(4-chlorophenyl)-4-(1H-pyrrole-3-carbonyl)morpholine
ethyl 1-ethyl-5-[(1-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(3,5-dimethoxyphenyl)methyl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
(1-{[5-(4-chlorophenoxy)-1,3-dimethyl-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)methanamine
(2S,4S)-N-ethyl-1-[(5-methylfuran-2-yl)methyl]-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
3-fluoro-N,5-dimethyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)imidazo[1,2-a]pyridine-2-carboxamide
(1R,5R)-6-[(3,4-dimethoxyphenyl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
9-(2-amino-6-methylpyrimidin-4-yl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N,6-dimethylpyrimidin-4-amine
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(3-phenylpiperidin-1-yl)acetamide
(1S,4S)-2-benzyl-5-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,5-diazabicyclo[2.2.1]heptane
5-(1-methyl-3-propyl-1H-pyrazol-5-yl)-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
5-(4-fluorophenyl)-N-[(1-methylpiperidin-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1,3,5-trimethyl-4-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}-1H-pyrazole
3-(2-amino-1,3-thiazol-4-yl)-N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]propanamide
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2-methyl-4-{4-[4-(pyridin-3-yl)piperazine-1-carbonyl]phenyl}butan-2-ol
2-{1-[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrrole-2-carboxamide
(1R,5R)-6-[(2,3-difluoro-4-methylphenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
methyl 6-({methyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]carbamoyl}amino)-1,2,3,4-tetrahydroquinoline-1-carboxylate
(2E)-1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
N-(1,3-benzothiazol-2-ylmethyl)-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
2-(1-methyl-1H-pyrrol-3-yl)-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]acetamide
(3aR,5R,6S,7aS)-2-{[5-chloro-2-(trifluoromethyl)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
N-{2-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}methanesulfonamide
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
2-(3-{1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}phenoxy)acetamide
2-[4-(2-methanesulfonamidoacetyl)morpholin-3-yl]-N-phenylacetamide
1-[4-({3-[3-(pyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)thiophen-2-yl]ethan-1-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidin-3-yl]methanol
6-[1-(morpholine-4-carbonyl)piperidin-4-yl]-2-(pyridin-2-yl)-3,4-dihydropyrimidin-4-one
N-[1-(methoxymethyl)cyclopentyl]-1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2S,4R)-1-(2-ethoxyacetyl)-N-ethyl-4-(4-fluoro-2-methylbenzamido)pyrrolidine-2-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}quinoline-3-carboxamide
N-(2-chlorophenyl)-3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propanamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-hydroxy-2-(pyridin-3-yl)ethyl]benzamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-(carbamoylmethyl)piperidine-4-carboxamide
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-(1H-imidazol-2-yl)benzamide
2-(piperidin-1-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
N-methyl-2-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2-(pyridin-3-yl)acetamide
7-(3-chlorophenyl)-4-(pyrrolidin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-1-(methoxymethyl)cyclobutane-1-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)oxan-4-amine