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N,1-dimethyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1H-imidazole-5-carboxamide
(3aS,6aS)-2-cyclopropanecarbonyl-5-(thiophene-2-sulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2,3-dimethoxyphenyl)methyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
1-(3-chlorophenyl)-4-[2-(methylamino)pyridine-4-carbonyl]piperazin-2-one
N-{[5-({ethyl[(4-ethylphenyl)methyl]amino}methyl)furan-2-yl]methyl}-N-methylmethanesulfonamide
1-cyclopropanecarbonyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxamide
3-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-methyl-5-phenyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-methyl-4-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
2-(4-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-2-oxopiperazin-1-yl)benzonitrile
2-{2-[4-(1H-pyrazol-1-yl)phenyl]phenyl}ethan-1-amine
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-[5-(4-methylphenyl)furan-2-yl]propan-1-one
1-(4-{[3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2-oxazol-5-yl]methoxy}phenyl)ethan-1-one
N-[2-(4-methoxyphenyl)ethyl]-5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
2-(4-chlorophenyl)-N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-hydroxyacetamide
N-(1-benzylpyrrolidin-3-yl)-3-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]propanamide
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{[(oxan-4-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N-cyclopropyl-5-[3-(1H-pyrazol-3-yl)phenyl]furan-2-carboxamide
4-(1H-1,3-benzodiazole-2-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
4-[(6-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}pyridin-3-yl)methyl]morpholine
N-(2-methoxyethyl)-3-{[1-(1-phenoxypropan-2-yl)piperidin-4-yl]oxy}benzamide
1'-(1H-indol-2-ylmethyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
5-fluoro-2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(pyrrolidin-1-yl)pyrimidine
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(thiophen-2-ylmethyl)piperazine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methyl-N-(quinoxalin-2-ylmethyl)acetamide
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one
(3aS,6aS)-2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{[3-(2-amino-1,3-thiazol-4-yl)propyl]sulfamoyl}-N-cyclopropylbenzamide
(2,1,3-benzoxadiazol-5-ylmethyl)[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
N-methyl-2-phenyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
4-{4-[2-(3-fluorophenyl)acetyl]piperazin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-methyl-3-{methyl[(4-pentylphenyl)carbamoyl]amino}propanamide
N-(3-hydroxy-3-methylbutyl)-N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
9-[2-(3,4-dimethylphenyl)acetyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
[(2-ethylpyrimidin-5-yl)methyl]({[2-(morpholin-4-yl)pyridin-3-yl]methyl})amine
2-acetyl-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(2R,4S)-4-hydroxy-1-[(2-methylnaphthalen-1-yl)methyl]piperidine-2-carboxylic acid
N2-(6-methoxypyrimidin-4-yl)-N1-(pyridin-3-yl)ethane-1,2-diamine
4-benzyl-1-(thiophene-2-carbonyl)-1,4-diazepan-5-one
dimethyl({3-[2-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-1H-imidazol-1-yl]propyl})amine
2-(2-methylphenyl)-5-{[4-(3-methylpyridin-4-yl)piperazin-1-yl]methyl}pyrimidine
1-ethyl-5-{1-[3-(methylsulfanyl)propyl]-4-phenyl-1H-imidazol-5-yl}-1H-1,2,4-triazole
1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
4-(4-benzylpiperazin-1-yl)-2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-[3-(2-fluorophenoxy)azetidine-1-carbonyl]pyridin-2-ol
4-(5-{[2-methyl-4-(2-methylphenyl)piperazin-1-yl]methyl}pyrimidin-2-yl)morpholine
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-[(2E)-but-2-en-1-yl]-5-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3,4-oxadiazole