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1-(2-hydroxyacetyl)-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
4-[4-({8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)phenyl]-2-methylbutan-2-ol
3-{methyl[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]amino}propan-1-ol
N-cyclohexyl-3-{[3-(piperidin-3-yl)phenyl]formamido}propanamide
2-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]benzoic acid
3-(2-{6-azabicyclo[3.2.1]octan-6-yl}-2-oxoethyl)-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
5-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
methyl 4-{[(2-{5-oxo-1-[1-(thiophen-2-yl)ethyl]pyrrolidin-2-yl}ethyl)amino]methyl}benzoate
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-1-propyl-1H-pyrazole-5-carboxamide
1-(4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)imidazolidine-2,4-dione
N-benzyl-N-methyl-2-(pyrimidin-5-yl)quinoline-4-carboxamide
2-(5-methyl-2-oxo-5-phenylpiperidin-1-yl)-N-(propan-2-yl)acetamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,3,4,7-tetramethyl-1H-indole-2-carboxamide
N-(3,5-dimethoxyphenyl)-3-[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-yl]propanamide
{5-[(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)methyl]-2-(propan-2-yloxy)phenyl}methanol
N-[2-hydroxy-3-(4-methylphenoxy)propyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
2-ethyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}pyrimidine
[(3R,5R)-1-(1,3-benzothiazole-5-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
(3S,4R)-1-[(5-methylfuran-2-yl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-ethyl-3-(morpholine-4-carbonyl)-N-[(1-phenylcyclopentyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)azepan-4-amine
methyl 4-{[(2S,4R)-2-{[(4-methylphenyl)methyl]carbamoyl}-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidin-1-yl]methyl}benzoate
1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
2-hydroxy-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-4-(methylsulfanyl)butan-1-one
2-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-methylthieno[3,2-d]pyrimidin-4-amine
(2S,4R)-4-[2-(carbamoylamino)acetamido]-N-ethyl-1-(2-phenylethyl)pyrrolidine-2-carboxamide
N-(5-hydroxypentyl)-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
[(3aS,6aS)-2-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
2-{1-[(3,4-difluorophenyl)methyl]-4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)propanamide
N-(furan-2-ylmethyl)-1,3-dimethyl-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
9-[(2-fluoro-4-methoxyphenyl)methyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(4aR,8aR)-7-[(3-chloro-4-methoxyphenyl)methyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)-5-(pyridine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[4-(aminomethyl)phenyl]methyl}-4-propylpyrimidine-5-carboxamide
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-3,5-dimethyl-1,2-oxazole
{4-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]morpholin-2-yl}methanamine
8-chloro-3-(2,2,6,6-tetramethylpiperidin-4-yl)-3,4-dihydroquinazolin-4-one
2-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]piperidin-1-yl}-1,3-benzoxazole
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-[4-(3-methylphenoxy)piperidin-1-yl]-3-(morpholin-4-yl)butan-1-one
2-{1-[(2-fluorophenyl)methyl]-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(1S)-1-[1-(2,5-dichlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethan-1-ol
8-[(2,5-difluorophenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(2-phenyl-1H-imidazol-1-yl)acetamide
N-(prop-2-en-1-yl)-2-(4-propanoylphenoxy)-N-(pyridin-2-ylmethyl)acetamide
N-methyl-1-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperidine-2-carboxamide
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-methyl-1-[3-(methylsulfanyl)phenyl]urea