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1-[(2,2-dimethyloxan-4-yl)methyl]-4-(2-methylpyridin-4-yl)piperazine
2-(2-methoxyethyl)-9-[2-(1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(3-ethylphenoxy)-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}azetidine
N-[(3R,4S)-4-cyclopropyl-1-(3-methylbutanoyl)pyrrolidin-3-yl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-2-(pyrrolidin-1-yl)acetic acid
[(1-methyl-1H-imidazol-2-yl)methyl]({[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl})(propan-2-yl)amine
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
7-(1-benzyl-1H-pyrazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-2,1,3-benzoxadiazole
2-(2-methyl-1,3-thiazol-4-yl)-1-[3-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
6-{4-[1-(2-methylphenyl)piperidin-4-yl]piperazin-1-yl}pyridine-3-carbonitrile
1-(1,3-benzothiazol-5-yl)-3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-methylurea
ethyl[(3-methyl-1,2-oxazol-5-yl)methyl][(trimethyl-1H-pyrazol-4-yl)methyl]amine
5-{[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
5-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole
7-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-4-(quinoxalin-5-ylmethyl)-1,4-diazepan-2-one
6-[3-(1H-pyrazol-3-yl)phenyl]pyrazolo[1,5-a]pyrimidine-2-carboxylic acid
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanamide
6-[3-(2,6-dimethylphenoxy)azetidin-1-yl]pyridine-3-carboxylic acid
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-methyl-N-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}propanamide
methyl 3-[(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)carbamoyl]propanoate
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-3-phenyl-1H-pyrazole-4-carboxamide
1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-N-[(4-methoxyphenyl)methyl]piperidine-4-carboxamide
5-(2,6-dimethoxyphenyl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1,2,4-triazin-3-amine
4-(4-chlorophenyl)-N-[(2S)-1-hydroxybutan-2-yl]butanamide
N-(3-fluorophenyl)-4-{[4-(2-hydroxypropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)propanoyl]piperazin-2-one
2-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]-1H-1,3-benzodiazole
9-[2-(morpholin-3-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
4-{[2-(3-fluorophenyl)-3-oxopiperazin-1-yl]methyl}benzamide
N,3-dimethyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-[2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-N,N-dimethylpyridine-3-carboxamide
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-sulfonyl}-3,5-dimethyl-1-phenyl-1H-pyrazole
1-(piperidin-1-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}cyclohexane-1-carboxamide
N-benzyl-2-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]acetamide
6-ethyl-N4-[(4-methoxypyridin-2-yl)methyl]-5-methylpyrimidine-2,4-diamine
1-{2-[(4aS,8aR)-1-(3-methylbutyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-chloro-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)pyridine-2-carboxamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(pyridin-2-yl)pyrimidine
3-butyl-4-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]-1-methylpiperazin-2-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-{[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amino}pyridine-3-carboxamide
3-(5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1,2,4-oxadiazol-3-yl)pyridazine
4-(5-{2-methyl-2,8-diazaspiro[4.5]decane-8-carbonyl}-1H-pyrazol-3-yl)phenol
N-({1-[(3S,5S)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)-N,4-dimethylpiperazine-1-carboxamide
2-fluoro-5-(6-methylquinolin-5-yl)benzamide
(benzylsulfamoyl)[2-(morpholin-4-yl)ethyl]amine
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-3-phenylpiperidine
N4-[1-(3-methylpyridin-2-yl)propan-2-yl]-6-(morpholin-4-yl)pyrimidine-2,4-diamine