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5,7-dimethyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)pyrido[2,3-d]pyrimidin-4-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
6-fluoro-8-[5-(methanesulfonylmethyl)pyridin-2-yl]quinoline
7-(cyclopropylmethyl)-2-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
7-(5-chloropyridin-2-yl)-4-[2-(1H-imidazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-chlorophenoxy)pyridine-3-carboxamide
1-benzoyl-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methylpiperidin-4-amine
1-[(3-methoxyphenyl)methyl]-3-phenyl-6-(1,3-thiazole-5-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(3-methylbut-2-enoyl)piperidine-2-carboxamide
3-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-1,3-diazinane-2,4-dione
3-[(3-aminopiperidin-1-yl)methyl]-N-[4-methyl-1-(2-methylpropyl)-1H-pyrazol-5-yl]benzamide
5-(4-cyclohexylphenyl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1,2,4-triazin-3-amine
1-(6-hydroxy-1,4-oxazepan-4-yl)-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propan-1-one
(1R,3S)-3-(2-aminoethoxy)-7-[4-(methylsulfanyl)benzoyl]-7-azaspiro[3.5]nonan-1-ol
1-(phenylcarbamoyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
methyl 9-(oxan-2-ylmethoxy)-7-oxo-3-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[3-(1H-pyrazol-1-yl)phenyl]-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
4-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
4-(4-{3-azaspiro[5.5]undecan-9-yl}piperazin-1-yl)-6-methylpyrimidin-2-amine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(3-methoxypropyl)-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
1-{3-[4-(6-ethylpyrimidin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
4-(1-{[(2-ethyl-2H-1,2,3-triazol-4-yl)carbamoyl]methyl}-1H-indazol-5-yl)-N,N-dimethylbenzamide
14-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
5-{[5-(2-fluoro-6-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-4-methyl-1,2,3-thiadiazole
6-methyl-2-phenyl-N-[1-(pyridin-2-yl)propyl]pyrimidin-4-amine
N-[2-(dimethylamino)ethyl]-1-methyl-N-[(4-methylphenyl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-methyl-N-[2-(2-methylphenyl)-1-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}ethyl]cyclobutanecarboxamide
1-methyl-N-[2-(piperidin-1-yl)butyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
1-[4-(furan-2-carbonyl)piperazin-1-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
N-(2-hydroxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
3-(2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
4-(1-benzyl-5-{[2-(difluoromethoxy)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)morpholine
3-({3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}methyl)-N-methyl-1,2,4-oxadiazole-5-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-3-{[(2-methylphenyl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
1-ethyl-N-[(2-methoxyphenyl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[1-(1H-indol-2-yl)ethyl]-N,5,6-trimethylpyridine-3-carboxamide
3-[(2-fluorophenyl)methoxy]-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}azetidine
2-({[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
N-[(3,4-difluorophenyl)methyl]-3-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}propanamide
[1-(4-chlorobenzoyl)-3-[(4-fluorophenyl)methyl]piperidin-3-yl]methanol
4-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-6-methoxypyrimidin-2-amine
2-cyclohexyl-N-{2-[4-(4-methyl-1,4-diazepane-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}acetamide
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-4-methyl-1,2,5-oxadiazole-3-carboxamide
5-ethyl-5-{1-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
(2-ethoxy-5-{[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]methyl}phenyl)methanol
3-ethyl-N-(2-methoxyethyl)-N-[(4-methoxyphenyl)methyl]-1H-pyrazole-5-carboxamide