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6-(2,5-dimethylfuran-3-yl)-2-(piperidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-(1-benzofuran-2-ylmethyl)-4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(1,3-thiazol-2-yl)ethyl]benzamide
N-[(2-ethoxy-3-methoxyphenyl)methyl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
4-{4-[(2-methoxypyridin-3-yl)methyl]piperazin-1-yl}-2-methyl-6-propylpyrimidine
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]pyridine-2-carbonitrile
2-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,4-dihydroquinolin-4-one
1-(oxolan-2-ylmethyl)-1-(pyridin-2-ylmethyl)-3-[3-(4H-1,2,4-triazol-4-yl)phenyl]urea
1-[(1-phenylcyclopropyl)methyl]piperidin-4-ol
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[(2E)-3-phenylprop-2-en-1-yl]-8-{spiro[2.3]hexane-1-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
3-{1-[2-(hydroxymethyl)phenyl]-1H-1,3-benzodiazol-2-yl}propan-1-ol
4-(2-methylfuran-3-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
methyl 6-{[butyl(methyl)amino]methyl}-3-(2-chloro-6-fluorobenzamido)thieno[2,3-b]pyridine-2-carboxylate
(4aS,7aR)-1-[2-(3-fluorophenyl)ethyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{1-[(2-ethoxyphenyl)methyl]-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
1-[2-(dimethylamino)-4-[(thiophen-3-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
3-[4-(2-methyl-1-benzofuran-5-carbonyl)piperazin-1-yl]-1,2-benzothiazole
2-(2-chloro-4-fluorophenoxymethyl)-N-(3-hydroxybutyl)-1,3-oxazole-4-carboxamide
N-{[1-(dimethylamino)cyclohexyl]methyl}-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-N-(2-methoxy-5-methylphenyl)piperidine-1-carboxamide
3-({[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[(1-ethylpyrrolidin-2-yl)methyl]-1H-pyrazole-4-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-4-(pyridin-3-yl)pyrimidin-2-amine
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine
2-[4-({2,5-dimethyl-3-[(4-methylpiperidin-1-yl)methyl]phenyl}methyl)piperazin-1-yl]acetamide
2-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-hydroxyquinoline-6-carboxamide
4-(2-methoxy-5-methylphenyl)-5-propylpyrimidine
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[2-(3-methylpyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
1-(2,5-dimethylbenzenesulfonyl)-3-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
N-[(5-methylfuran-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-(1H-indol-3-yl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)ethan-1-one
8-[2-(1,2-benzoxazol-3-yl)acetyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(furan-2-yl)ethyl]-3-phenylpropanamide
N,N-dimethyl-4-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}aniline
N-(1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
methyl 5-[(4-hydroxybutan-2-yl)amino]-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}-2,6-dimethylphenol
N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[3-(3-methylpyrazin-2-yl)-1H-pyrazol-1-yl]acetamide
[5-({4-[4-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)furan-2-yl]methanol
N-methyl-5-(morpholin-4-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-oxazole-3-carboxamide
2-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(2R,3R,6R)-5-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[5-(cyclohex-3-ene-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
2-ethyl-6-methyl-5-{2-oxo-2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
5-tert-butyl-4-{[2-(4-fluorophenyl)morpholin-4-yl]methyl}furan-2-carboxamide
N-(2-propanoyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-4-(trifluoromethyl)benzamide