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N-(3-{4-[(thiophen-2-ylmethyl)amino]piperidin-1-yl}phenyl)pyridine-3-carboxamide
11-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
1-{4-[2-(4-methylpentyl)morpholine-4-carbonyl]phenyl}pyrrolidin-2-one
2-[(3-chlorophenyl)methyl]-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-[(2-propylpyrimidin-5-yl)methyl]piperidin-3-amine
N,6-dimethyl-N-(oxolan-3-ylmethyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-[(1R,9aR)-octahydro-1H-quinolizine-1-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-cyclohexyl-3-(cyclopropylmethyl)-N,N-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]azepan-4-amine
9-[(3-ethoxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-2H-1,3-benzodioxole-5-carboxamide
3-[(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidin-1-yl)methyl]pyridine
N-(3-{[(2-fluoroethyl)carbamoyl]methoxy}phenyl)propanamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-acetamidobutanoyl)pyrrolidine-3-carboxylic acid
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl){[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}amine
3-[(4aR,7aS)-4-(2-ethylbenzoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
(1R,2R,6S,7S)-4-(3-propyl-1H-pyrazole-4-carbonyl)-4-azatricyclo[5.2.1.02,6]decane
N-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
(3aR,6aR)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N,5-dimethylpyrazine-2-carboxamide
N-(1-methoxybutan-2-yl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
4-[2-(1-benzofuran-2-yl)-5-fluoropyrimidin-4-yl]morpholine
[benzyl(methyl)sulfamoyl][(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]amine
2,6-dimethyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}quinoline-4-carboxamide
2-{[3-(ethylcarbamoyl)pyrrolidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-amino-8-hydroxy-4-(oxolan-3-yl)-5H,6H-benzo[h]quinoline-3-carbonitrile
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
N-(1-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(2-methoxyphenyl)acetamide
1-[(diethylcarbamoyl)methyl]-N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-methoxy-1-{4-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
2-methyl-1-(1,3-thiazol-5-ylmethyl)-1,4-dihydroquinolin-4-one
4-[2-(2,3-dimethoxyphenyl)acetyl]-1-(4-methylphenyl)piperazin-2-one
N-(3,4-dimethoxyphenyl)-2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-methoxy-1-{4-[4-(3-propanoylpiperidine-1-carbonyl)phenoxy]piperidin-1-yl}propan-1-one
2-(2-aminoethyl)-N-(2-methoxyethyl)-N-(3-phenylprop-2-yn-1-yl)quinazolin-4-amine
N-(2-{3-cyclopropyl-1-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}ethyl)-N-methylmethanesulfonamide
(3S,4S)-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
3-{[1-(2H-1,3-benzodioxol-5-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(piperidin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
5-[4-(4-chlorophenyl)piperazine-1-carbonyl]-1-cyclohexyl-N-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]urea
1-benzyl-N3-cyclopropyl-N5-[2-(1H-indol-3-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(1-cycloheptylpiperidin-3-yl)ethyl]piperidine-4-carboxamide
3-[(3R,4S)-1-{2-amino-6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-(carbamoylmethyl)-N-[(5-methoxy-1H-indol-2-yl)methyl]piperidine-4-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazole
3-[(3-fluorophenyl)methyl]-5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
N-[(3R,5S)-5-(diethylcarbamoyl)-1-propanoylpyrrolidin-3-yl]pyrazine-2-carboxamide
1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-4-carboxamide