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1-(2-cyclopropylphenyl)-3-[1-(morpholin-4-ylmethyl)cyclopentyl]urea
4-(3-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-yl}propoxy)benzamide
6-oxo-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,6-dihydropyridazine-3-carboxamide
3-(3-hydroxyazetidine-1-carbonyl)-1-methyl-1,2-dihydroquinolin-2-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]acetamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-methyl-1-[(5-methylfuran-2-yl)methyl]-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
8-(4-hydroxy-3-methylbenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[3-(difluoromethyl)-5-methyl-1H-pyrazol-1-yl]-1-[4-(4-fluorophenoxy)piperidin-1-yl]ethan-1-one
3-(3-fluorophenyl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]benzamide
7-(2-hydroxyethyl)-2-[4-(1H-pyrazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butane-1,2-dione
2-(2-chloro-4-fluorophenoxymethyl)-N-[1-(5-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
2-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1,3-thiazole-4-carboxamide
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-pentyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
dimethyl({5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]furan-2-yl}methyl)amine
2-[5-(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
ethyl 4-(3-aminoazepan-1-yl)piperidine-1-carboxylate
(3S,4S)-1-[3-(furan-2-yl)propanoyl]-4-propylpyrrolidine-3-carboxylic acid
2-{2-[4-(oxan-4-yl)piperazin-1-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-(1,4-oxazepan-4-yl)butan-1-one
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]oxolane-2-carboxamide
2-[({1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
4-phenyl-1-[6-(pyridin-4-yl)pyridine-3-carbonyl]azepane
1,3-dimethyl 5-{[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]amino}benzene-1,3-dicarboxylate
1-[(3-fluoro-4-methoxyphenyl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]thiophene-3-carboxamide
4-[1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]benzoic acid
(2-{3-[3-(4-methanesulfonylphenyl)phenyl]-1H-pyrazol-1-yl}ethyl)dimethylamine
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)[(2,4,5-trimethylphenyl)methyl]amine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-cyclohexyl-N-ethyl-1H-pyrazole-4-carboxamide
N-benzyl-5-{1-[(1-methylpyrrolidin-3-yl)methyl]-1H-imidazol-2-yl}pyrimidin-2-amine
N-methyl-2-propyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyridine-4-carboxamide
2-amino-1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-methylpropan-1-one
ethyl 4-[7-(1H-inden-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
1-cyclohexanecarbonyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrrolidine-2-carboxamide
3-({[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazol-5-yl]formamido}methyl)benzoic acid
1-(4-chlorophenyl)-N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]cyclobutane-1-carboxamide
6-{[4-(hydroxymethyl)phenyl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-(2-{[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
3-ethyl-1-[1-(4-methoxyphenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]urea
1-(1,4-dioxan-2-ylmethyl)-5-(1-methylcyclopropyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
N-(1-methanesulfonylpiperidin-4-yl)-2-methyl-5-propylpyrimidin-4-amine
(3aS,6aS)-5-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-N,N-dimethyl-octahydropyrrolo[3,4-b]pyrrole-1-carboxamide
(3S,4R)-1-(1-benzofuran-5-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-2-one
3-chloro-5-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-amine
2-(3-hydroxyphenyl)-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}acetamide
(2R,3R)-3-amino-1'-(isoquinoline-1-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol