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1-(9H-fluoren-2-yl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
1-(cyclohexylcarbamoyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[2-(2-oxopiperidin-1-yl)ethyl]benzamide
1,3-dimethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(5-methyl-1,3,4-thiadiazol-2-yl)-3-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carboxamide
1-(3-chloro-4-methoxyphenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-oxopyrrolidine-3-carboxamide
1-[(4-fluorophenyl)methyl]-3-({[(3-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
8-(4-aminopiperidine-4-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}-2-[4-(1H-pyrazol-5-yl)phenyl]acetic acid
4-(3-hydroxyphenyl)-N-(2-methyl-1H-1,3-benzodiazol-6-yl)piperidine-1-carboxamide
1-(6-hydroxy-1,4-oxazepan-4-yl)-3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
6-[2-(2-methoxyphenyl)ethyl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2-(propan-2-ylsulfanyl)acetamide
ethyl 4-[(4-chlorophenyl)methyl]-1-(3-phenoxypropanoyl)piperidine-4-carboxylate
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(2-methylphenyl)methyl]piperidin-4-ol
2-{[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
propan-2-yl (4aS,7aR)-6,6-dioxo-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
3-(5-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
3-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-7-methoxy-1-(prop-2-yn-1-yl)-1,2-dihydroquinolin-2-one
8-[(2S,4S)-4-amino-1-methylpyrrolidine-2-carbonyl]-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethoxy)ethan-1-one
(1R,5R)-3-(3-chloro-4-fluorobenzoyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-cyclopropyl-9-(2-hydroxyethyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-methyl-5-{2-[2-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3S,7S)-5-(2-ethylpyridine-4-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
ethyl 1-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
N-(2-cyano-3-methylphenyl)-3-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}benzamide
1-benzyl-8-[1-(methylsulfanyl)propan-2-yl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4S)-1-[(4-hydroxyphenyl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
N5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N5,N6,N6-trimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
6-(methoxymethyl)-2-(3-{[methyl(1,2,3,4-tetrahydronaphthalen-1-yl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[2-(pyridin-3-yloxy)ethyl]acetamide
ethyl 1-{[5-(methoxymethyl)furan-2-yl]methyl}-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
[(3R,4R)-1-(2-chloro-5-methylbenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-hydroxy-N-methyl-2-(3-methylphenyl)pyrimidine-5-carboxamide
N-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
N-methyl-2-(methylamino)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-thiazole-4-carboxamide
6-methyl-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
4-(4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)-2-methylbutan-2-ol
3-(3-fluorophenyl)-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1H-pyrazole
N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[2-(dimethylamino)ethyl]-N-ethyl-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(2-oxopyrrolidin-1-yl)acetamide
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
1-[(3S,4R)-1-(2,5-dimethylfuran-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}quinoline-3-carboxamide
N-methyl-N-(oxan-4-ylmethyl)-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide