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N4-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-(6-cyclopropylpyrimidin-4-yl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylic acid
5-ethyl-1'-(quinoline-6-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(3-fluorophenyl)ethyl]-5-{4-hydroxy-1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}-1-benzofuran-2-carboxamide
4-hydroxy-2-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrimidine-5-carboxamide
4-[(4-fluorophenyl)methyl]-1-(3-hydroxypyridine-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-{4-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]phenyl}pyrrolidin-2-one
7-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidine
1-propyl-5-[3-(1H-pyrazol-5-yl)phenyl]-1H-1,2,4-triazole
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(2,4-dimethylphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-hydroxy-3-({[(2-methylpyridin-4-yl)methyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
3-(5-aminopentyl)-5-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
methyl(2-phenylethyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
5-({3-[2-(1-benzofuran-2-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)pyrimidine
6-(3-chloro-4-methoxyphenyl)pyrazine-2-carboxylic acid
[7-(2,6-dimethylpyridin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methanamine
2-methoxy-N-[(2R,3R)-1'-[5-(methoxymethyl)thiophene-2-carbonyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-benzyl-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
N-(pyridin-4-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-amine
2-(3-methylthiophene-2-carbonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(quinoline-3-carbonyl)pyrrolidin-3-yl]methanol
1-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}butan-2-ol
7-[(4-fluorophenyl)methyl]-2-(3-methylbutanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}-1-propyl-1H-pyrazole-5-carboxamide
1-[6-(3-{[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyridin-3-yl]ethan-1-one
4-[4-(2-butylpyrrolidine-1-carbonyl)phenyl]-2-methylbutan-2-ol
5-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-5-ethyl-3-[2-(4-methoxyphenyl)ethyl]imidazolidine-2,4-dione
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(2H-indazol-2-yl)-N-methylacetamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
3-(1H-indol-3-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}propanamide
1-{4-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)urea
N-{2-methyl-4-[methyl(pyridin-2-ylmethyl)carbamoyl]phenyl}furan-2-carboxamide
2-ethoxy-3-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]pyridine
N-{[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
3-({7,9-dioxo-8-azaspiro[4.5]decan-8-yl}methyl)benzonitrile
1-{5-[5-(3-ethyl-5-methyl-1,2-oxazol-4-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
2-(ethylsulfanyl)-5-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)pyrimidine
3-({[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]amino}methyl)phenol
2-{2-[1-(2,6-dimethoxypyridine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
3-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)propanoic acid
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}ethane-1-sulfonamide
1-methyl-8-[3-(5-methylfuran-2-yl)butyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 3-[(2,4-difluorophenyl)methyl]-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-3-carboxylate
4-benzyl-3-ethyl-1-(1-propyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
3-{[(furan-3-ylmethyl)amino]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
2-(naphthalen-1-yl)pyridine-3-carboxylic acid
ethyl[(3-fluoro-2-methylphenyl)methyl][(1-methyl-1H-imidazol-2-yl)methyl]amine
N-butyl-3-{[2-(hydroxymethyl)-2,5-dihydro-1H-pyrrol-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide