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N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-3-(propylamino)-5-(pyrrolidine-1-sulfonyl)benzamide
2-cycloheptyl-1-{4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
ethyl 4-(8-fluoro-4-oxo-1,4-dihydroquinoline-3-amido)piperidine-1-carboxylate
methyl 3-[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})carbamoyl]benzoate
4-(4-chlorophenyl)-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(6-methoxypyrimidin-4-yl)piperidin-3-ol
5-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}-1H-1,3-benzodiazole
2-amino-5-methyl-4-[3-(morpholin-4-ylmethyl)phenyl]-6-phenylpyridine-3-carbonitrile
(1S,5R)-6-[(5-methylthiophen-2-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-hydroxy-4-methylbenzamide
N-{4-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-3-methylphenyl}acetamide
(1S,5R)-6-benzyl-3-[(2,3-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(2-{1-[(2-methoxy-4-methylphenyl)methyl]piperidin-3-yl}ethyl)acetamide
3-chloro-4-fluoro-N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
1-methyl-N-[2-(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]piperidine-3-carboxamide
3-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]-N-[(2-methoxyphenyl)methyl]propanamide
2-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-6-methyl-4H-pyran-4-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-5-phenyl-1,2-oxazole-3-carboxamide
2-hydroxy-N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]pyridine-3-carboxamide
1-[1-(methoxymethyl)cyclopentyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
8-(4-methyl-1,3-thiazole-5-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(5S)-5-{[({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(pyridin-4-ylmethyl)amino]methyl}pyrrolidin-2-one
3-amino-1-[(2-cyclohexylpyrimidin-5-yl)methyl]pyrrolidine-3-carboxylic acid
(1S,5R)-3-cyclobutanecarbonyl-N-(3,5-dimethylphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
7-(1,3-benzothiazole-6-carbonyl)-2-oxa-7-azaspiro[4.5]decane
1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(5-methylpyrazin-2-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
methyl 4-(5-{[methyl(quinoxalin-6-ylmethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
4-{[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}benzoic acid
N,1-dimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N,4-dimethyl-3-(2-oxoimidazolidin-1-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
N-(3-methanesulfonamidophenyl)-7-methoxy-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-[(3,4-dimethylphenyl)methyl]-4-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]piperazin-2-one
5-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-4-ethyl-1,3-thiazol-2-amine
2-{[2-(dimethylamino)ethyl](methyl)amino}-6-[4-(methylsulfanyl)phenyl]-N-(thiophen-2-ylmethyl)pyridine-3-carboxamide
1-[4-(dipropylamino)piperidin-1-yl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
3-[4-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]pyrrolidin-2-one
1-methyl-2-(morpholin-4-yl)-N-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
2-[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-5-methyl-2,3-dihydro-1H-indole
1-{[(3R,4R)-1-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
(2E)-3-(2-fluorophenyl)-1-(4-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)prop-2-en-1-one
3-benzyl-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]-1-methyl-2,3-dihydro-1H-indol-2-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(morpholin-3-yl)acetamide
3-(1H-indol-3-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]propanamide
2-[3-(dimethylamino)propyl]-9-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-methyl-1-benzofuran-5-carboxamide
N-ethyl-2-{3-[3-(4-methoxypyrimidin-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
4-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}morpholine