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(3R,5S)-N3-methyl-N3-[(3-methyl-1,2-oxazol-5-yl)methyl]-N5-(4-methylphenyl)piperidine-3,5-dicarboxamide
1-(2-methyl-6-propylpyrimidin-4-yl)-N-(oxan-4-yl)piperidin-4-amine
[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]diphenylmethanol
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
2-(4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
methyl[(1S)-1-[3-(oxan-4-yl)-1-propyl-1H-1,2,4-triazol-5-yl]pentyl]amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[4-(pyrimidin-2-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]acetamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-2-methyl-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(4-chloro-3-fluorophenyl)methyl]piperazin-2-one
1-{1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]piperidin-3-yl}pyrrolidin-2-one
2-(ethylamino)-N-[2-(phenylsulfanyl)ethyl]-N-(prop-2-en-1-yl)pyrimidine-5-carboxamide
5-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazin-2-ol
[(3R,4R)-1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
2-[3-(1H-imidazol-1-yl)propyl]-N-[(2R)-3-methylbutan-2-yl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-4-(piperidin-1-yl)butanamide
4-[1-(4-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}phenyl)ethyl]morpholine
N-[2-(pyridin-3-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
6-(propan-2-yloxy)-N4-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrimidine-2,4-diamine
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-phenyl-1,4-diazepane
2-[1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
2-[(1S,4S)-5-(2-methoxy-5-phenylphenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]-N,N-dimethylacetamide
2-amino-1-(4-{[4-(thiomorpholin-4-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)propan-1-one
N-[(7-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]furan-2-carboxamide
N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
[(4-ethynylphenyl)methyl](2-methoxyethyl)(thiophen-2-ylmethyl)amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-4-(1H-pyrazol-1-yl)benzamide
1-(2-methoxypyridine-4-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-methyl-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}propanamide
(2R)-2-amino-3-hydroxy-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
1-(4-ethylpiperazin-1-yl)-3-[3-({[(1-methylpiperidin-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
7-fluoro-N-methyl-N-(2-methylpropyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
2-{5-[4-(4-methylpiperazin-1-yl)phenyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]pyridin-2-amine
methyl 5-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-(2-fluorophenyl)piperidin-4-amine
8-(4,6-dimethoxypyrimidin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N,8-dimethyl-4-oxo-N-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}-1,4-dihydroquinoline-3-carboxamide
5-{[8-(3-hydroxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-N,N-dimethylfuran-2-carboxamide
2-[(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)oxy]-4-methoxy-N-(2-methoxyethyl)benzamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1,5-dimethyl-1H-indazole-3-carboxamide
1-{4-[(2,1,3-benzoxadiazol-5-ylmethyl)amino]-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-benzyl-N3-[(1-hydroxycyclohexyl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(3,4-dimethoxyphenyl)methyl](2-methoxyethyl)amine
2-(2-methoxy-5-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(2-methyl-1,3-thiazol-4-yl)-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrimidin-4-ol
2-(2,4-dichlorophenoxy)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
2-chloro-N-(1-{1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide