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1-[5-(methoxymethyl)furan-2-carbonyl]-4-(2-methoxyphenoxy)piperidine
1-{3-[({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)amino)methyl]phenyl}ethan-1-one
6-methoxy-3-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1-benzofuran-2-carboxamide
2-amino-4-[4-methoxy-3-(methoxymethyl)phenyl]-6-propyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(3S,4S)-1-ethyl-4-methoxypyrrolidin-3-yl]-2,7,8-trimethylquinoline-4-carboxamide
N-ethyl-N-methyl-6-[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]pyridine-3-carboxamide
3-{1-[2-(azepan-1-yl)acetyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[4-(quinolin-8-yl)-1H-pyrazol-1-yl]acetamide
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(methylsulfanyl)pyrimidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
6-ethyl-2-[4-({4-[2-(1H-imidazol-1-yl)ethyl]piperazin-1-yl}methyl)phenyl]-3,4-dihydropyrimidin-4-one
7-(3-methoxypropanamido)-N-(thiophen-2-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-{4-[(3-phenylpropyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
5-(1H-indol-3-ylmethyl)-1-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole
2-methyl-5-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,4-dihydropyridin-4-one
N-ethyl-N-methyl-6-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidin-4-amine
3-(2-carbamoylphenyl)benzoic acid
1-({1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
1-[2-methyl-2-(piperidin-1-yl)propyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-cyclopropyl-2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)acetamide
3-ethyl-8-[3-(2-oxoimidazolidin-1-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1-(propan-2-yl)piperidine
7-chloro-4-hydroxy-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]quinoline-3-carboxamide
(3S,4S)-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
4-{5-[(4-methoxy-2,3-dimethylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-1H-pyrazole
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N,5-dimethyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
N,N-dimethyl-2-{[3-(thiophen-3-yl)propanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
5-({[(3-{2-[4-(3-fluorobenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
{2-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}urea
N-cyclopropyl-1-ethyl-3-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
2-[N-(3-fluorophenyl)methanesulfonamido]-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]acetamide
3-(1-butyl-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazole-3-carbonyl)piperidine
2-[2-oxo-2-(2-phenylmorpholin-4-yl)ethyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-ol
1-(5-tert-butyl-2-methoxyphenyl)-3-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]urea
4-(3,5-dimethyl-1-benzofuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 4-[3-hydroxy-3-(hydroxymethyl)piperidine-1-carbonyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
3-(5-{[(2R,6S)-2,6-dimethylpiperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridazine
4-[7-(3-ethoxypropanoyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
1-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
[(2,6-difluoro-3-methoxyphenyl)methyl][3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]methylamine
1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-4-(pyridin-3-yl)piperazine
3-[1-(3-chloro-2-methylphenyl)-1H-imidazol-2-yl]pyridine
4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-(6-methyl-1H-1,3-benzodiazol-7-yl)benzamide
(1S,5R)-3-(pyrazine-2-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{1-oxa-8-azaspiro[4.5]decan-8-yl}-2-(3-phenylpyrrolidin-1-yl)ethan-1-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-difluoro-6-methoxybenzamide
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide