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3-cyclopropyl-6-(3-methanesulfonylphenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
3-[(dimethylamino)methyl]-1-{[3-(2-methylpropoxy)phenyl]methyl}piperidin-3-ol
2,5-dioxo-6-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-2-(piperidin-1-ylmethyl)-1,4-oxazepane
(3R,4S)-4-cyclopropyl-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-amine
N-(4-chloro-3-methoxyphenyl)-2-[(1,1-dioxo-1λ6-thiolan-3-yl)(prop-2-en-1-yl)amino]acetamide
methyl (2S,4S,5R)-4-[(2-ethoxy-2-oxoethyl)(methyl)carbamoyl]-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylate
2-methyl-N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)-1,3-thiazole-4-carboxamide
1-(5-{[4-(1,3-benzothiazol-2-yl)-1,4-diazepan-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
3-{2-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-2-methyl-1,4-dihydroquinolin-4-one
4-(azocane-1-sulfonyl)-N-(2-hydroxyethyl)benzamide
N-(cyclohexylmethyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-6-methyl-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
benzyl(methyl){[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidine-3-carboxamide
2-[3-({5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}methyl)phenoxy]acetamide
2-{4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]morpholin-3-yl}-1-(2,5-dihydro-1H-pyrrol-1-yl)ethan-1-one
4-(1-methyl-1H-indol-2-yl)-3-(propan-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
(4aS,8aR)-6-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
3-methyl-6-{5-[(3-methylphenyl)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
4-[(3-methyl-3-phenylpiperidin-1-yl)sulfonyl]morpholine
4-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-1-(4-methylphenyl)piperazin-2-one
3-(4-chlorobenzoyl)-1-[3-(methylsulfanyl)propyl]piperidine
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2-cyclohexyl-1,3-benzoxazole-6-carboxamide
6-{2-[(4-methoxyphenyl)methoxy]phenyl}pyrimidin-4-amine
1-({4-[(2R,5R)-2,5-dimethylpyrrolidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
2-[(quinolin-4-ylmethyl)(thiophen-2-ylmethyl)amino]butan-1-ol
2-methyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-5-(propan-2-yl)furan-3-carboxamide
5-{[2-(1-propylpiperidin-3-yl)ethyl]carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
2-[(1-ethyl-1H-indol-3-yl)sulfanyl]-1-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
N-methyl-1-(2-phenylethyl)-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}piperidin-4-amine
N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
6-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
1-(oxan-4-yl)-N-{3-[(pyridin-3-yl)amino]propyl}piperidine-3-carboxamide
ethyl 5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-methylbutanamide
1-(4-methoxyphenyl)-3-methyl-4-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}piperazin-2-one
methyl[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]{[2-(propan-2-yl)pyrimidin-5-yl]methyl}amine
3-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}pyridin-2-ol
5-(1-benzofuran-2-yl)-1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazole
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-1H-pyrazole-4-carboxamide
1-[4-(1H-imidazol-1-yl)phenyl]-3-methyl-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}urea
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[(4-acetamidophenyl)methyl]piperidine-3-carboxylate
8-{[3-(2-aminoethyl)phenyl]methyl}-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{2-[5-(2,2-dimethyloxan-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}propanamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[3-(pyridin-4-yl)propyl]acetamide