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1-{2-[4-(3-chloro-5-fluoro-4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-(1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)pyridine
N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-oxo-1,2-dihydroquinazoline-4-carboxamide
(4aR,8aR)-4a-hydroxy-7-[3-(hydroxymethyl)-8-methylquinolin-2-yl]-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
2-(1H-pyrazol-1-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]butan-1-one
N-[4-(1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1H-1,2,3-triazol-4-yl)phenyl]acetamide
2-{[(2-fluoro-3-methoxyphenyl)methyl](methyl)amino}-N,N-dimethylpropanamide
2-benzyl-9-(2-ethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,5R)-N-phenyl-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-(cyclohex-3-en-1-yl)-1-(2-propoxyethyl)-1H-1,2,3-triazole
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-2-(trifluoromethyl)benzene-1-sulfonamide
N-[2-({[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}amino)ethyl]methanesulfonamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
(2E)-3-(4-methoxyphenyl)-1-{4-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}prop-2-en-1-one
1-ethyl-N-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
1-[3-(1H-pyrazol-1-yl)benzoyl]-4-(4H-1,2,4-triazol-4-yl)piperidine
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(2-hydroxyethyl)-N-(1-phenylethyl)-5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-methoxy-5-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)benzoic acid
N-[2-(4-{[benzyl(methyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]thiophene-3-carboxamide
1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-3-(pyrazin-2-yl)propan-1-one
3-{2-[methyl(2-methylpropyl)amino]ethyl}-8-(1,3-thiazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1,4-dioxan-2-ylmethyl)-N-methyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
(3S,4R)-4-(4-fluorophenyl)-1-{[2-(2-hydroxyethoxy)phenyl]methyl}pyrrolidine-3-carboxylic acid
1-[(1-hydroxycyclohexyl)methyl]-3-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-(1H-pyrrole-2-carbonyl)piperazine
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
5-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-5-oxopentanamide
1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-methoxypiperidine
(2S,4R)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-hydroxypyrrolidine-2-carboxamide
N,3,5-trimethyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
(2S,4R)-N-ethyl-4-[(1-ethylpiperidin-4-yl)amino]-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
[1-(2-methoxyphenoxy)propan-2-yl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
1-{2-[(2-methylpropyl)amino]benzoyl}piperidine-4-carboxylic acid
4-methoxy-N-{[1-(pyridin-4-yl)piperidin-3-yl]methyl}benzene-1-sulfonamide
4-ethyl-3-[(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-methyl-2-{4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidin-4-amine
(2S,4R)-4-hydroxy-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxamide
3-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-5-(propan-2-yl)-1,2,4-oxadiazole
(1S,5R)-3-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{1-[(1-propyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}benzonitrile
2-ethyl-N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)butanamide
(3aS,6aS)-2-(cyclopropylmethyl)-1-oxo-5-[3-(pyridin-3-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-5-(naphthalen-2-yl)-1,2,4-triazin-3-amine
3-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-1-(thiophen-2-yl)urea
{3-[(dimethylamino)methyl]-1-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperidin-3-yl}methanol
ethyl[(1-methyl-1H-imidazol-2-yl)methyl]({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amine
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-[(1-phenylcyclopentyl)methyl]piperidine-3-carboxamide
methyl 4-({4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carbonyl}amino)benzoate
2-amino-7-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one