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2-[3-oxo-9-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(1-phenyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methanol
N-ethyl-2,6-dimethoxy-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrimidine-4-carboxamide
5-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-1-(2-ethoxyethyl)-4-phenyl-1H-imidazole
(1S,5R)-N-(3,4-dimethylphenyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-{4-[2-(4-fluorophenyl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
N-ethyl-2-{[2-(1-hydroxycyclopentyl)ethyl](methyl)amino}pyridine-3-carboxamide
N-cyclopentyl-N'-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}butanediamide
2-[3-(2,5-dimethoxyphenyl)-1H-pyrazol-1-yl]-N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]acetamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl){[5-(methoxymethyl)furan-2-yl]methyl}amine
(3aS,6aR)-5-(furan-3-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-({1-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
2-{3-[(1-methylpiperidin-4-yl)methyl]-5-(2-phenylpropyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
5-(3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)pyrimidine
7-(2-phenylquinazolin-4-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-1,3-thiazol-4-yl)methanol
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]amino}methyl)piperidin-2-one
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(ethyl)(oxolan-2-ylmethyl)amine
N-{1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
N-[(3-chlorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]spiro[2.2]pentane-1-carboxamide
N-({1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}methyl)-4-fluorobenzamide
{1-[1-(4,6-dimethylquinazolin-2-yl)piperidin-4-yl]piperidin-4-yl}(thiophen-2-yl)methanol
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-(2-methylpyridin-4-yl)piperazine
methyl 4-[4-(1-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)piperazin-1-yl]benzoate
[(2-{5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}phenyl)methyl]dimethylamine
8-(3-acetylbenzoyl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-8-methyl-2-(thiophen-2-yl)quinoline
N-[(3R,4S)-1-(2-amino-2-methylpropyl)-4-propylpyrrolidin-3-yl]furan-2-carboxamide
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxybenzoyl)piperazine
2-(2,3-difluorophenyl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]-1-(2-methylpropyl)piperidin-4-amine
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-2,2,6,6-tetramethylpiperidin-4-amine
1-[2-(1-methylpyrrolidin-2-yl)ethyl]-2-[4-(methylsulfanyl)phenyl]-1H-imidazole
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl){[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}amine
1-ethyl-4-{[4-(4-methoxyphenoxy)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N,N-diethyl-3,6-dimethyl-2-(1-propyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[1-({3-[6-oxo-4-(pyridin-4-yl)-1,6-dihydropyrimidin-2-yl]phenyl}methyl)pyrrolidin-3-yl]acetamide
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
2-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)pyridine-3-carboxamide
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-hydroxypropan-1-one
N-(1-{1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
5-{5-[3-(1H-indol-3-yl)propyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
4-chloro-N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-methyl-1H-indole-2-carboxamide
(3R,4R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
1-cyclopropyl-N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1H-pyrrole-2-carboxamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-(3-hydroxypropyl)-N-(thiophen-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[(1S)-1-(4-chlorophenyl)ethyl]-4-[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-3-methylpiperidine