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8-(1H-indol-2-ylmethyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
4-{[1-(3-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
N-{1-[1-(adamantan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-amine
1-methyl-4-{3-[2-(methylsulfanyl)ethyl]-5-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl}piperidine
4-{2-[2-(1-ethyl-1H-1,2,4-triazol-5-yl)-1H-imidazol-1-yl]ethyl}benzene-1-sulfonamide
N-(2-{[(2-chloro-3-methoxyphenyl)carbamoyl]amino}ethyl)acetamide
2-[4-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
1-{2-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
methyl 5-(cyclohexylamino)-3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1,3-dimethyl-4-[6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carbonyl]piperazin-2-one
1-{5-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl}butan-2-ol
8-[2-(4-phenylpiperidin-1-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(4-{[1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)acetic acid
2-(3-methoxypropyl)-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-(2-fluorophenyl)-4-{[4-(4-methylpiperidine-1-carbonyl)-1,3-oxazol-2-yl]methyl}piperazine
2-(cyclopropylmethyl)-9-(2,3-difluoro-4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-({[(1-ethyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amino}methyl)benzonitrile
N-(2-methoxyethyl)-N-methyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
4-(pyridin-3-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-2-amine
2-methoxy-N-[1-methyl-2-phenyl-5-(4-phenylpiperidine-1-carbonyl)-1H-1,3-benzodiazol-7-yl]acetamide
1-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazole-2-carbonyl}piperidine-4-carboxamide
3-[3-({[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
3-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(2-methoxyethyl)[(4-methylphenyl)methyl]amino]propane-1,2-diol
(2S)-2-{[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]formamido}propanamide
(3aS,6aR)-5-(6-methoxypyrimidin-4-yl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(2,2-diphenylethyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
5-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-chloro-6-methyl-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-(adamantan-1-ylmethyl)-N-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(2-chlorophenyl)-2-{[4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethan-1-ol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
1-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-4-(hydroxymethyl)azepan-4-ol
3-phenyl-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
5-({8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-2-(pyridin-2-yl)pyrimidine
1-(4-fluorophenyl)-4-(oxolan-3-ylmethyl)-1,4-diazepane
5-(3-fluoro-4-methoxybenzenesulfonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
5-[(2E)-but-2-en-1-yl]-N-(isoquinolin-5-ylmethyl)-N-methyl-1,3,4-oxadiazole-2-carboxamide
4-[3-(4-methyl-1,4-diazepan-1-yl)propanoyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
(4aS,7aR)-1-(5-chloropyridine-2-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cyclohexyl-3-(cyclopropylmethyl)-5-(5-oxo-1,4-diazepane-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-(3-carbamoyl-4-methoxyphenyl)azocane-1-carboxamide
3-(1-{1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
N-methyl-9-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-N,N-diethylpyrrolidin-3-amine
3-(4-methoxyphenyl)-5-(thiophene-3-sulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-6-(piperidin-3-yl)pyrimidin-4-amine
(2S,4S)-1-benzyl-4-{[(2,6-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide