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3-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]benzonitrile
3-(3,5-difluorophenyl)-5-(morpholine-4-sulfonyl)benzoic acid
1-[(4aR,8aR)-7-cyclopentanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-(thiophen-2-yl)ethan-1-one
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]urea
N-[(3S,4R)-1-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-pyrazol-1-yl)propan-1-one
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-cyclopentylpropan-1-one
8-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-(dimethylamino)-2-(3-methylphenyl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-N-(2-phenylethyl)-2-(thiomorpholine-4-carbonyl)-2,3-dihydro-1H-inden-2-amine
1-ethyl-6-{[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-indole
(1R,3S)-3-(2-hydroxyethoxy)-7-(1H-imidazol-2-ylmethyl)-7-azaspiro[3.5]nonan-1-ol
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(3-hydroxyphenyl)piperazin-1-yl]ethan-1-one
8-(7-fluoro-2-methylquinoline-4-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-cyclopropyl-1-{2-[1-(4-fluorobenzoyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-methyl-4-(3-methyl-1H-pyrazol-1-yl)benzoic acid
2-(adamantan-1-yl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-3-carboxamide
3-(oxolan-3-yl)-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1,2,4-oxadiazole
5-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-amine
6-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-5,6-dihydro-1,6-naphthyridin-5-one
2-(pyridin-2-yl)-7-(1H-pyrrole-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6-fluoro-2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-1H-1,3-benzodiazole
({4-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(pyridin-4-ylmethyl)amine
3-{[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]sulfamoyl}-N,N-dimethylbenzamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
1-cyclopropyl-4-[4-(pyridin-4-ylmethyl)piperazine-1-carbonyl]pyrrolidin-2-one
1-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
(3S,4S)-1-(4-methoxybenzoyl)-4-[methyl({[3-(methylsulfanyl)phenyl]methyl})amino]pyrrolidin-3-ol
8-[(2,5-difluorophenyl)methyl]-3-ethyl-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{3-[6-(propan-2-yloxy)pyridazin-3-yl]phenyl}methanol
5-({[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]amino}methyl)pyrimidin-2-amine
2-methyl-2-[4-(morpholin-4-yl)-2-(3,3,4-trimethylpiperazin-1-yl)pyrimidin-5-yl]propanoic acid
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}amine
1-(3,5-dimethylphenyl)-4-(4-methyl-1,3-thiazol-2-yl)piperazin-2-one
1-(propan-2-yl)-2-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
N-(2,1,3-benzoxadiazol-4-ylmethyl)-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
2-(2-{2-[2-(methylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)-1,2,3,4-tetrahydrophthalazine-1,4-dione
3-[(diethylamino)methyl]-N-[2-(hydroxymethyl)phenyl]benzamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-4-oxo-1,4-dihydroquinoline-2-carboxamide
4-(5-methylpyridin-2-yl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-4-ol
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]thian-4-amine
6-{[3-(benzyloxy)phenyl]methyl}-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
methyl (2S,4R)-1-(quinolin-4-ylmethyl)-4-{2-[3-(trifluoromethyl)phenyl]acetamido}pyrrolidine-2-carboxylate
1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
N-ethyl-N-methyl-2-{3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-8-yl}acetamide
2-[4-(4-fluorophenoxy)piperidin-1-yl]-2-(6-methoxypyridin-3-yl)acetic acid