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N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}-2-(2-oxopiperidin-1-yl)acetamide
7-[(5-phenylthiophen-2-yl)methyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
9-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(3-fluorophenyl)ethyl]-2-(4-{4-[(furan-2-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
3-(3-methoxyphenyl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
6-chloro-3-(1,3-dihydroxypropan-2-yl)-8-methyl-3,4-dihydroquinazolin-4-one
4-({4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]furan-2-yl}methyl)morpholine
[7-(4-chloro-1-methyl-1H-indazol-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-3,5-dimethyl-1H-indole
(2S)-3-hydroxy-2-(methylamino)-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}propanamide
6-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridine-6-carbonyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-ethyl-3-(2-methylpropyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-pyrazole-5-carboxamide
7-methyl-3-[(5-phenylthiophen-2-yl)methyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
3-[(3R,4S)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-[(4-fluorophenyl)methyl]-5-hydroxy-N-(oxolan-2-ylmethyl)pyrazine-2-carboxamide
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-2-(3-hydroxyadamantan-1-yl)acetamide
3-{2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propyl}pyridine
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-2-propoxyethan-1-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(2-methylpyridin-4-yl)methyl]acetamide
N-tert-butyl-1-cyclohexyl-4-oxo-5-(4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-{2-[(1-cyclopentylpiperidin-3-yl)formamido]ethyl}pyridine-3-carboxamide
N-cyclopropyl-1-[1-(2-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-5-(methoxymethyl)thiophene-2-carboxamide
6-ethyl-4-{[(pyridin-4-ylmethyl)amino]methyl}-2H-chromen-2-one
2-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}pyridine-4-carbonitrile
1-[(3,4-difluorophenyl)methyl]-3-{[ethyl(methyl)amino]methyl}-3-hydroxypiperidin-2-one
5-(2-chloro-4-fluorophenoxymethyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,2-oxazole-3-carboxamide
5-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane-2-carbonyl)pyridin-2-ol
4-(2,5-dimethylpyrimidin-4-yl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-cyclohexyl-N-(2-hydroxy-2-phenylethyl)-2-methyl-1,3-thiazole-4-carboxamide
1-benzyl-N-[(3-methylpyridin-4-yl)methyl]-4-phenylpiperidine-4-carboxamide
2-(5-methyl-1H-pyrazol-1-yl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-[(4-methylphenyl)sulfanyl]-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
(3S,5R)-5-[(6-methylpyridin-3-yl)carbamoyl]-1-[(3-methylthiophen-2-yl)methyl]piperidine-3-carboxylic acid
3-{4-[4-(trifluoromethyl)piperidin-1-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl}-1H-indole
2-(2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-oxoethoxy)acetamide
2-methyl-2-{[2-(1H-pyrazol-1-yl)phenyl]formamido}propanamide
(4-phenylbutan-2-yl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
5-butyl-1'-(5-methylthiophene-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(piperidin-1-yl)-1-(1H-1,2,3-triazole-5-carbonyl)piperidine-4-carboxamide
2-{8-methyl-2,8-diazaspiro[4.5]decane-2-carbonyl}-N-(pyridin-2-ylmethyl)aniline
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-(trifluoromethyl)benzamide
5-[(adamantan-2-ylmethyl)amino]-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-({4-[(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amino]-6-methylpyrimidin-2-yl}amino)phenol
[1-(1H-1,3-benzodiazol-2-yl)ethyl]({[7-chloro-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
N-cyclopropyl-4-({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}sulfamoyl)benzamide
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}oxolane-3-carboxamide