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1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-3-(dimethylamino)pyrrolidine-1-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[2-(dimethylamino)ethyl]-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(pyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N'-(4-methoxyphenyl)-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]propanediamide
2-(2,5-dimethylphenoxy)-N-(furan-3-ylmethyl)propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-3-ol
2-{1-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]azetidin-3-yl}pyridine
3-cyclopropyl-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
4-{4-[(2-hydroxyphenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-4-oxo-3,4-dihydroquinazoline-2-carboxamide
3-{2-[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-ethyl-4-hydroxy-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-methylphenyl)pyrimidine-5-carboxamide
(2S,4R)-N,N-diethyl-4-(2-hydroxyacetamido)-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
4-methyl-2-{2-oxo-2-[2-(trifluoromethyl)pyrrolidin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-{4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]morpholin-3-yl}acetamide
8-(1,3-benzothiazol-2-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[2-(1H-pyrazol-1-yl)ethyl]-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
(2S,4S,5R)-4-{[(1-ethyl-1H-imidazol-2-yl)methyl]carbamoyl}-5-(2-fluorophenyl)-1-methylpyrrolidine-2-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-N-(1-hydroxybutan-2-yl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
(2S,4R)-N,N-diethyl-1-propyl-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-amido}pyrrolidine-2-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
5-hydroxy-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}pyrazine-2-carboxamide
3-chloro-4-({1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
N-cyclopropyl-3-[1-(2,2,2-trifluoroethanesulfonyl)piperidin-4-yl]propanamide
[1-({[2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}methyl)cyclopentyl]methanol
3-[1-(1-methyl-1H-indazol-5-yl)-1H-imidazol-2-yl]phenol
N-(3-cyano-4-methoxyphenyl)-4-[(3-fluorophenyl)methyl]-1,4-diazepane-1-carboxamide
2-({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(ethyl)amino)ethan-1-ol
N-cyclobutyl-3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)propanamide
1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
(3aR,6aR)-2-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}-1-[(4-ethoxyphenyl)methyl]piperidin-4-ol
(1R,3S)-3-(3,3-diphenylpiperidine-1-carbonyl)cyclopentan-1-amine
1-{2-hydroxy-3-[4-methoxy-2-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
N-(3,4-dimethylphenyl)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
4-(azepan-1-ylmethyl)-N-(4H-1,2,4-triazol-4-yl)benzamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
N-[1-(pyridin-2-yl)propan-2-yl]-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amine
2-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
1-[(2,4-difluoro-3-methoxyphenyl)methyl]-4-(oxan-4-yl)piperazine
5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-2-(methoxymethyl)pyrimidine
2-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-N-[5-(ethylsulfanyl)-1,3,4-thiadiazol-2-yl]acetamide
1-(furan-2-ylmethyl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
1-{1-[(4-ethynylphenyl)methyl]piperidin-3-yl}-4-(2-fluorophenyl)piperazine
4-{[(3R,4S)-3-cyclobutaneamido-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-N-methylbenzamide
(1R,3S)-7-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-7-azaspiro[3.5]nonane-1,3-diol
(3aS,6aR)-5-(1,4-dithiepan-6-yl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one