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2-[(3,5-difluorophenyl)methyl]-8-(1,4-dioxan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
[1-(1-methyl-1H-pyrazol-4-yl)ethyl]({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
(3S,4R)-N,N-dimethyl-1-(1-methyl-1H-indole-3-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-amine
3-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridazine
2-(4-chlorophenyl)-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]morpholine
2-[4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)phenyl]acetamide
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-hydroxypropan-1-one
2-[5-cyclopropyl-4-(4-ethylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(2-fluorophenyl)pyrimidine
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
2-(2,5-dimethoxyphenyl)-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}acetic acid
3-[(2-fluorophenyl)formamido]-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)propanamide
1-(4-{[(2R,5S)-5-[(3-fluoro-4-methylphenyl)methyl]oxolan-2-yl]methyl}piperazin-1-yl)ethan-1-one
(1R,5R)-6-(cyclobutylmethyl)-3-(5-methylpyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(4aR,6R,8aS)-2-[(2-ethyl-1,3-thiazol-4-yl)methyl]-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
2-(4-fluorophenyl)-4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}morpholine
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-3-carboxamide
3-(4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]acetamide
N-(3-chloro-4-propanamidophenyl)-2-propyl-1,3-thiazole-4-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-[3-(thiophen-2-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
2-methyl-4-[4-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}methyl)phenyl]butan-2-ol
[(3-fluoro-4-methoxyphenyl)methyl]({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)amine
(3R,5S)-N-(2,3-dihydro-1H-inden-5-yl)-1-(2-methylpropyl)-5-(piperidine-1-carbonyl)piperidine-3-carboxamide
2-(4-methylpentyl)-4-(propane-1-sulfonyl)morpholine
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[2-(phenylsulfanyl)ethyl]piperidine
2-{4-[(5-methylthiophen-2-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
ethyl 3-[({1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}carbamoyl)amino]propanoate
methyl 3-[(2E)-3-(2-chlorophenyl)prop-2-enamido]-5-{[(4-methyl-1H-imidazol-2-yl)formamido]methyl}benzoate
4-phenyl-1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}azepane
6-oxo-1-(2-phenylethyl)-N-[2-(pyrazin-2-yl)ethyl]piperidine-3-carboxamide
(1S,5R)-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]-N-(pyridin-4-ylmethyl)quinoline-4-carboxamide
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}amine
3-(3-fluorophenyl)-N-[1-(1,3-thiazol-2-yl)propyl]-1H-pyrazole-4-carboxamide
2-(2,4-dichlorophenoxy)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}acetamide
1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(thian-4-yl)piperazine
(3R,4R)-N,1-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(2-methyl-1H-imidazol-5-yl)pyrrolidine-3-carboxamide
1-(2-fluorophenyl)-4-[4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]piperidin-4-ol
N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-4-(thiophene-2-carbonyl)piperazine-1-carboxamide
5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-phenyl-1H-imidazole
6-(cyclopropylmethyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-5,6-dimethylpyridine-3-carboxamide
5,7-dimethyl-N-[2-methyl-1-(4-methylpiperazin-1-yl)propan-2-yl]pyrido[2,3-d]pyrimidin-4-amine
4-[(1E)-3-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}prop-1-en-1-yl]-2-methoxyphenol
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[6-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]propan-1-ol
3-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
({4-[(5-ethylpyridin-2-yl)methyl]-1,4-oxazepan-6-yl}methyl)dimethylamine
N-[4-(2-hydroxy-3-methylbutanamido)phenyl]-5-methylfuran-3-carboxamide
3-fluoro-5-[1-(2-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]benzonitrile