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N-[2-(2-fluorophenoxy)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
4-(1-methyl-1H-pyrazol-4-yl)-1-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]-1,2,3,6-tetrahydropyridine
4-{[(4aR,8aR)-4a-hydroxy-7-(2-methoxyacetyl)-decahydro-2,7-naphthyridin-2-yl]methyl}benzoic acid
[2-(azepan-1-yl)ethyl](ethyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
1-[5-(oxolan-2-yl)thiophene-2-carbonyl]-4-(1H-pyrrole-2-carbonyl)piperazine
3-ethyl-N-[2-methyl-3-(pyrrolidine-1-carbonyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
N-[2-(furan-2-yl)ethyl]-4-(morpholine-4-sulfonyl)benzamide
1-{4-[(dipropylamino)methyl]benzoyl}piperidine-3-carboxylic acid
N-ethyl-N-[2-(3-methylphenoxy)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(4-hydroxyphenyl)benzamide
4-{[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
2,4-dimethyl-N-{2-[methyl(phenyl)carbamoyl]phenyl}pyrimidine-5-carboxamide
1-(2-methoxyphenyl)-4-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}piperazin-2-one
4-[3-(2-methoxybenzoyl)piperidin-1-yl]-6-(methoxymethyl)pyrimidine
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-(2,3,6-trimethylphenoxy)ethan-1-one
2-methyl-3-{3-[1-(prop-2-en-1-yl)-1H-pyrazol-3-yl]phenyl}pyrazine
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]thiophene-3-carboxamide
9-{[4-(2-aminoethyl)phenyl]methyl}-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-({8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}methyl)-1H-pyrazole-3-carboxylate
N-phenyl-5-[3-(phenylamino)piperidine-1-carbonyl]pyrimidin-2-amine
N-{imidazo[1,2-a]pyrazin-3-ylmethyl}pyrazine-2-carboxamide
methyl 2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetate
(2R)-1-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}pyrrolidine-2-carboxamide
4-(2,4-dimethylbenzoyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
1'-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-(2-methoxyphenyl)-4-[4-(pyrrolidin-1-yl)pentanoyl]piperazin-2-one
3-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}propanamide
{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}[(4-methyl-1H-imidazol-5-yl)methyl]amine
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-(2-phenylethyl)-1H-pyrazole-4-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(phenylformamido)acetamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(pyrimidin-4-ylmethyl)benzamide
6-methoxy-N-methyl-N-[2-(phenylsulfanyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1R,5S,6S)-3-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-N-methyl-3-azabicyclo[3.1.0]hexane-6-carboxamide
(3S,4S)-1-{[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
1-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
5-(2-phenoxyethyl)-3-(2-phenylethyl)-1H-1,2,4-triazole
2-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]-4,6-dimethylpyridine-3-carbonitrile
2-{1-[(2-ethoxyphenyl)methyl]-4-(pyridine-2-carbonyl)piperazin-2-yl}ethan-1-ol
8-[(2-fluoro-5-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-3-ol
1-[(3-chlorophenyl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
5-[1-(2,5-dimethylpyrimidin-4-yl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
4-[(4-methyl-5-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
2-(1-butyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
1-(5-acetylpyridin-2-yl)-4-(3-tert-butyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-[4-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)piperidin-1-yl]pyridine-3-carbonitrile
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-(4-methanesulfonylphenyl)-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
3-{4-[3-(methylsulfanyl)propyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one