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1,7-dimethyl-5-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-2,4-dione
ethyl 4-{[1-(6-chloropyridazin-3-yl)piperidin-4-yl]amino}piperidine-1-carboxylate
4-ethyl-3-(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,4-dimethyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
(3aS,6aR)-5-(4,6-dimethoxypyrimidin-2-yl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(3R,4S)-4-cyclopropyl-1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]-1H-1,2,3-benzotriazole-5-carboxamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
3-ethyl-8-[2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4R)-4-amino-1-(3,4-dihydro-2H-1,5-benzodioxepine-7-sulfonyl)-N-methylpyrrolidine-2-carboxamide
1-{1-[(5-chlorothiophen-2-yl)methyl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-(oxan-3-yl)pyridin-2-amine
2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-[(1S)-1-phenylethyl]acetamide
2-{4-[(3-ethoxy-4-methoxyphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
N-cyclopropyl-2-({1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
N3-{2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-N1-(pyridin-3-yl)propane-1,3-diamine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
6-(2-aminoethyl)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-methylpyrimidin-4-amine
N-benzyl-N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
1-[2-(dimethylamino)ethyl]-3-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-3-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(3-fluoro-4-methoxyphenyl)-3-(piperidine-1-carbonyl)pyridine
N-methyl-5-({methyl[2-(morpholin-4-yl)ethyl]amino}methyl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[2-(dimethylamino)ethyl]-1-[1-(2-fluorophenyl)piperidin-4-yl]-N-methylpiperidin-3-amine
1-(azocan-1-yl)-3-[2-methoxy-5-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
1-(2-methoxyacetyl)-N-[2-(quinolin-8-yloxy)ethyl]piperidine-3-carboxamide
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(1-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carbonyl}piperidin-4-yl)methanol
(3S,4R)-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-(1-{1-[(5-fluoro-2-methoxyphenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
4-ethyl-3-({1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-methyl-2-[(4-methylpiperazin-1-yl)methyl]quinolin-4-ol
4-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}pyridine
methyl 2-(1H-1,3-benzodiazol-5-ylformamido)-2-(3-methylphenyl)acetate
1-({4-methyl-5-[1-(1,3-thiazol-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
5-(2-fluoro-4,5-dimethoxyphenyl)-4-phenyl-1-[2-(pyrrolidin-1-yl)ethyl]-1H-imidazole
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
{[4-(cyclopentyloxy)phenyl]methyl}(1H-imidazol-2-ylmethyl)methylamine
3-methyl-1-(3-methylphenyl)-5-[(trimethyl-1H-pyrazol-1-yl)methyl]-1H-1,2,4-triazole
5-{1-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazol-4-yl}-2-chloropyridine
3-methyl-8-[4-(1,3-oxazol-5-yl)benzenesulfonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(1,2-thiazole-5-carbonyl)pyrrolidin-3-yl]methanol
4-[(4-fluorophenyl)methyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-[2-(dimethylamino)ethyl]-3-methylthiophene-2-carboxamide
6-(4-fluorophenyl)-7-(3-methylbut-2-en-1-yl)-2-(2-methylpyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
methyl (2S)-1-{3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanoyl}pyrrolidine-2-carboxylate
2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-1,3-benzoxazole
5-methoxy-2-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-4H-pyran-4-one
N-cyclohexyl-3-[(5-methoxy-4-oxo-1,4-dihydropyridin-2-yl)formamido]propanamide
6-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}quinoline