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1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(3-methylpyridin-4-yl)-1,4-diazepane
2-acetyl-8-[3-(4-fluorophenoxy)propyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(3R,4S)-1-(4-aminopyrimidin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-3-methanesulfonylpropanamide
1-(butan-2-yl)-5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-N-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(1H-imidazol-2-yl)ethyl]-1,3-oxazole-4-carboxamide
6-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3,4-dihydropyrimidin-4-one
[1-(1-aminocyclopropanecarbonyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
1-(3-methoxypropyl)-3-[2-oxo-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-3-phenylpyrrolidine-2,5-dione
(4aS,8aR)-6-(4-methyl-1H-pyrrole-2-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-{3-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
3-({1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
3-{4-[(2-ethylpyrimidin-4-yl)methyl]piperazin-1-yl}-2,5-dimethylpyrazine
N'1-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopropane-1,1-dicarboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(5,6-dimethylpyrimidin-4-yl)piperazin-2-yl}ethan-1-ol
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(methylsulfanyl)ethan-1-one
2-(dimethylamino)-2-(2-fluorophenyl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
(benzylsulfamoyl)[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]amine
1-methyl-4-[(1-{[3-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]piperazine
7-(1-benzothiophen-3-yl)-4-(4-hydroxybutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{[3-(furan-2-yl)-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
2-amino-4-(3,4-dihydroxyphenyl)-5H-thiochromeno[4,3-b]pyridine-3-carbonitrile
1-{2-[(3-methylpyridin-4-yl)amino]ethyl}-3-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
4-({4-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]furan-2-yl}methyl)morpholine
(3aR,6aR)-2-[(3-chloro-2-fluorophenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-N-[2-(4-methoxyphenyl)ethyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-oxo-4H-chromene-2-carboxamide
6,6-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]-5-oxothiomorpholine-3-carboxamide
1-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-[9-(1-ethyl-1H-pyrazole-4-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
(1-{[2-(4-ethylphenyl)-1H-imidazol-1-yl]methyl}cyclobutyl)methanol
methyl (2R,4S)-4-hydroxy-1-{2-[(thiophen-2-ylmethyl)amino]benzoyl}piperidine-2-carboxylate
N-ethyl-2,4,5-trimethyl-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
N-[3-(dimethylamino)propyl]-2-{4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]morpholin-3-yl}acetamide
1-(pyridin-3-ylmethyl)-4-{[3-({1-[4-(trifluoromethoxy)benzenesulfonyl]piperidin-4-yl}oxy)phenyl]methyl}piperazine
4-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-5-oxopyrrolidine-3-carboxylic acid
N-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}-5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
4-(1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)thiomorpholine
8-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
6-{2-[(dimethylamino)methyl]phenyl}-N-(propan-2-yl)pyrimidin-4-amine
1-{2-[(2-aminopyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-2-phenoxyethan-1-one
1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
1-[(3-methoxyphenyl)methyl]-4-(quinolin-4-ylmethyl)piperazin-2-one
N-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-(pyridin-2-yl)azetidine-1-carboxamide
4-acetyl-N-[2-(morpholin-4-ylmethyl)phenyl]-1,4-diazepane-1-carboxamide
(4aS,8aR)-1-(3-aminopropyl)-6-[2-(benzyloxy)acetyl]-decahydro-1,6-naphthyridin-2-one
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)acetamide
3-hydroxy-3-({[2-(methylamino)ethyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
1-methyl-N-[2-(pyridin-4-yl)ethyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-ethyl-8-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione