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7-[1-(methoxymethyl)cyclobutanecarbonyl]-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-methyl-1-phenyl-4-(pyrimidin-5-yl)-1H-pyrazol-5-amine
N-[(2S,4R,6S)-2-{3-[(diethylamino)methyl]-4-methoxyphenyl}-6-ethyloxan-4-yl]acetamide
4-hydroxy-2-methyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-5-carboxamide
(2R,4S)-4-hydroxy-1-[2-(trifluoromethoxy)benzenesulfonyl]piperidine-2-carboxylic acid
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)pyrrolidine-1-carboxamide
2-[4-(1H-imidazol-1-yl)phenyl]-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-imidazole
2-methyl-5-{[3-(2-phenylethyl)piperidin-1-yl]methyl}-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-(5-fluoro-2-methyl-1H-indol-3-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)acetamide
3-(2-oxo-2-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)imidazolidine-2,4-dione
N-(2-propyl-2H-1,2,3-triazol-4-yl)-3-(1,2,3,6-tetrahydropyridin-1-ylmethyl)benzamide
1-benzyl-8-[4-(1H-indol-3-yl)butan-2-yl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2-(pyridin-3-yl)morpholine
8-(2,6-dimethylpyridin-4-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-{3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]propanoyl}-1-(3-chlorophenyl)piperazin-2-one
5-ethyl-2,3-dimethyl-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-(1H-1,2,3,4-tetrazol-1-yl)-1-[2-(thiomorpholin-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
4-ethyl-2-methyl-N-{3-[methyl(phenyl)amino]propyl}-1,3-thiazole-5-carboxamide
2-{3-[(2-methoxyphenyl)methoxy]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-fluoro-4-[4-(1H-pyrazol-5-yl)phenyl]benzene-1-sulfonamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
1,3-dimethyl-N-(oxan-4-yl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(4aS,8aR)-6-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
ethyl 1-(2-hydroxyethyl)-5-[3-(5-methylfuran-2-yl)butyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(2,6-dimethylpyridin-4-yl)piperazine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-methyl-1H-pyrazole-3-carbonyl)pyrrolidine-3-carboxylic acid
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-3-methylthiophene-2-sulfonamide
N-[2-(ethylsulfanyl)ethyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-{3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]morpholin-4-yl}-2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethan-1-one
N-{4-[(4-{4-[(propan-2-yl)amino]pyrimidin-2-yl}piperazin-1-yl)methyl]phenyl}acetamide
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-5-propyl-1,2-oxazole-3-carboxamide
9-[(4-chloro-3-fluorophenyl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[4-({ethyl[(3R,4R)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]amino}methyl)phenyl]acetamide
3-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridin-2-amine
N-[4-(3-fluorophenyl)phenyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)pyrrolidine-2-carboxamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-5-(oxolan-3-yl)-1H-1,2,4-triazol-3-yl]pyridine
3-(pentan-2-yl)-8-(1,3-thiazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{2-[4-(2,2-dimethylpropyl)morpholin-2-yl]ethyl}-1,2-oxazole-5-carboxamide
4-{[(1-methyl-1H-imidazol-2-yl)methyl]amino}-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
2-(dimethylamino)-N-[4-(1,2-oxazolidine-2-carbonyl)phenyl]acetamide
(4aS,8aR)-1-(4-hydroxybutyl)-6-(5-methoxyfuran-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-benzyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(2S,4S)-4-amino-1-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-{[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}pyridin-2-amine
3-(2-oxo-2-{1-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}ethyl)-2,3-dihydro-1H-isoindol-1-one
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propanoic acid
N-(1,2-oxazol-3-ylmethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide