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N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[4-(pyrimidin-4-yl)-1H-pyrazol-1-yl]acetamide
1-(4-methoxyphenyl)-2-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}-1H-imidazole
1-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(propan-2-yl)urea
5-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}propane-1-sulfonamide
3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
N-(2,2-difluoroethyl)-4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
4-[4-(2-methoxypyridin-3-yl)-2-methylquinolin-3-yl]butan-2-one
4-(2-oxopyrrolidin-1-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}benzamide
ethyl 3-[(2E)-3-phenylprop-2-en-1-yl]-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-3-carboxylate
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-(1,4-oxazepan-4-ylmethyl)piperidin-2-one
N,N-diethyl-1-{1-[2-(naphthalen-1-yl)acetyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl){[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}amine
N-(but-2-yn-1-yl)-1-[2-(3-fluorophenyl)ethyl]-N-(furan-2-ylmethyl)-6-oxopiperidine-3-carboxamide
3-({[2-(2,5-dimethylphenoxy)ethyl](methyl)amino}methyl)-1-methyl-1,2-dihydroquinolin-2-one
N-[2-(3-chlorophenoxy)ethyl]-N-ethyl-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
4-ethyl-3-{[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(butan-2-yl)(pyridin-4-ylmethyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]-N-[2-(hydroxymethyl)phenyl]benzamide
1,4-dimethyl 2-[(5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-1H-pyrazol-4-yl)formamido]butanedioate
1'-[3-(1H-imidazol-2-yl)benzoyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
N-[(3,4-difluorophenyl)methyl]-3-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-3-yl}propanamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
5-[(6-methoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
4-(5-{[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
1-(4-{4-azaspiro[2.5]octan-4-ylmethyl}phenoxy)-3-[benzyl(methyl)amino]propan-2-ol
(2S,4R)-4-(dimethylamino)-1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)pyrrolidine-2-carboxylic acid
2,4-dimethoxy-6-(2,3,4-trimethoxyphenyl)-1,3,5-triazine
4-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperazine-2-carboxylic acid
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-3-(thiophen-3-yl)propan-1-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
6,8-dimethyl-3-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)-1,2-dihydroquinolin-2-one
2-(thiophen-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,3-thiazole-4-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-benzothiophene-5-carboxamide
methyl (2S,4R)-4-(dimethylamino)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidine-2-carboxylate
(1S,5R)-3-(pyrazine-2-carbonyl)-N-(thiophen-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
3-[(3R,4S)-1-[4-(ethylamino)pyrimidin-2-yl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-{imidazo[1,2-a]pyridin-3-yl}-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)acetamide
4-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-N-methylpyridin-2-amine
5-tert-butyl-3-({4-propyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1H-pyrazole
1-ethyl-N-[(5-fluoro-1H-indol-2-yl)methyl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
7-(4-chloro-1-methyl-1H-indole-2-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
7-methoxy-3-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
8-[(3-hydroxyphenyl)methyl]-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3-hydroxypropyl)-1-{1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-(adamantan-1-yl)-4-(dimethyl-1,3-thiazole-5-carbonyl)piperazine
2-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
2-(benzyloxy)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one