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1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(4-methylphenoxy)ethan-1-one
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-6-(piperidin-4-yl)pyrimidin-4-amine
(4aS,7aR)-1-(2-ethylbenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[3-(cyclopropylmethyl)-1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl]methanol
7-[(2,3-dimethoxyphenyl)methyl]-2-[(5-methylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decane
13-(5-ethylfuran-2-yl)-4,6-dimethyl-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
9-(cyclopropylmethyl)-4-(1-ethylpiperidin-4-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(2-phenoxyethyl)-1,4-diazepan-5-one
{5-[(5-cyclohexylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
1-(1-phenoxypropan-2-yl)-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
3-hydroxy-3-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)-1-[(3-methylphenyl)methyl]piperidin-2-one
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}({imidazo[1,2-a]pyrimidin-2-ylmethyl})amine
6-[4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-2,3-dihydropyridazin-3-one
2-{[ethyl(4-hydroxybutyl)amino]methyl}-6-fluoroquinolin-4-ol
(3aS,6aS)-2-(furan-3-carbonyl)-5-[(2-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1R,7S)-N-methyl-3-[(3-methylphenyl)methyl]-4-oxo-N-(1H-pyrazol-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-[(1S,2R)-2-aminocyclobutyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
N,5-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-[(3-{pyrazolo[1,5-a]pyridin-3-yl}phenyl)methyl]morpholine
N,5-dimethyl-2-[(propan-2-yl)amino]-N-[2-(pyridin-2-yl)ethyl]benzamide
N-[2-(2-methylpropanesulfonyl)ethyl]pyrimidin-2-amine
1-(4-fluorophenyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1,4-diazepane
6-(2-methylpropyl)-2-oxo-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2-dihydropyrimidine-4-carboxamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]({[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})methylamine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-4-(pyridin-2-yl)pyrimidin-2-amine
N,2-diethyl-N-{[4-(methylsulfanyl)phenyl]methyl}pyrimidine-5-carboxamide
N-{2-[3-(thiomorpholin-4-ylmethyl)phenoxy]propyl}furan-2-carboxamide
3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-N-methylpyridin-2-amine
2-({[(1S,2S)-2-hydroxycyclohexyl]amino}methyl)-6-methylquinolin-4-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propanamide
4-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}-5-methylpyrimidine
2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(propan-2-yl)acetamide
4-[2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carbonyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
5-[4-(piperidine-1-carbonyl)phenyl]quinoline
4-hydroxy-N-methyl-2-[(phenylsulfanyl)methyl]-N-(thian-4-yl)pyrimidine-5-carboxamide
2-ethyl-4-methyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1,3-oxazole-5-carboxamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)piperidin-3-yl]propanoic acid
2-(benzyloxy)-1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]ethan-1-one
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)pyrrolidin-3-ol
3-(4-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)pyrazine-2-carbonitrile
8-{imidazo[1,2-a]pyridine-3-carbonyl}-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2-{2-[1-(2-ethylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
1-(carbamoylmethyl)-N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]piperidine-4-carboxamide
6-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-(3-{[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,4-triazol-5-yl)acetamide
3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-1-ethyl-4,6-dimethyl-1,2-dihydropyridin-2-one
1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-benzyl-4-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)piperazin-2-one