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5-(1H-1,3-benzodiazol-6-yl)-1,2,3,4-tetrahydroisoquinoline
2-butyl-8-(4-methyl-1H-imidazole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-tert-butyl-4-(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carbonyl)pyrrolidin-2-one
ethyl 4-[(4-chlorophenyl)methyl]-1-(3-acetamidopropanoyl)piperidine-4-carboxylate
{4-[(5-chlorothiophen-2-yl)methyl]-1,4-oxazepan-6-yl}methanol
4-methyl-6-{4-[3-(1H-pyrazol-1-yl)benzoyl]piperazin-1-yl}pyrimidin-2-amine
2-{4-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
1-methanesulfonyl-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1,4-diazepane
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-2-(dimethylamino)-2-(2-methylphenyl)acetamide
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
2-(4-chlorophenoxy)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]acetamide
[8-methyl-2-(1,2,3,4-tetrahydroisoquinolin-5-yl)quinolin-3-yl]methanol
3,5-dichloro-4-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}pyridine
4-[3-({4-[(dimethylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
1-{2,7-diazaspiro[4.5]decan-7-yl}-3-(3,4-dimethoxyphenyl)propan-1-one
9-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-({4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}methyl)-5-methyl-1H-indole
4-[(4-fluorophenyl)methyl]-1-(thiolan-3-yl)piperidine
3-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2,5-dimethyl-1-phenyl-1H-pyrrole
1-(2-methylpropyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
4-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
3-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-N-benzyl-N-(cyclopropylmethyl)-1,2-oxazole-5-carboxamide
2-methoxy-2-methyl-N-[(3R,4S)-1-methyl-4-phenylpyrrolidin-3-yl]propanamide
5-(4-methylphthalazin-1-yl)pyridin-3-amine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenylpyrrolidin-2-one
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-methyl-1-(2-methyl-1-benzofuran-7-yl)urea
N-[3-(4-ethylpiperazin-1-yl)propyl]pyrimidin-2-amine
1,4,6-trimethyl-3-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-[3-(2-amino-1,3-thiazol-4-yl)propyl]-5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methylpiperidin-2-one
4-(3-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propyl)piperazin-2-one
2-methyl-1-[4-(morpholin-4-yl)benzoyl]piperidine-2-carboxylic acid
4-{5-[5-(ethoxymethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}pyrimidin-2-amine
1-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}-4-(methoxymethyl)piperidine
2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}-2-(thiophen-3-yl)acetic acid
6-methoxy-2-oxo-N-[3-(pyridin-3-yloxy)propyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-(methanesulfonylmethyl)piperidine
3-(2,5-dimethoxyphenyl)-5-(1H-pyrazol-3-yl)-1,2,4-oxadiazole
6-fluoro-2-[(3-hydroxyazetidin-1-yl)methyl]quinolin-4-ol
ethyl 4-({[4-(1H-1,2,4-triazol-1-yl)phenyl]carbamoyl}amino)piperidine-1-carboxylate
1-(2-methoxyethyl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(2,6-difluorobenzoyl)pyrrolidine-3-carboxylic acid
2-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-1,3-thiazole-4-carboxamide
N-[4-(3-methoxyphenyl)phenyl]-1-[2-(methylsulfanyl)acetyl]pyrrolidine-2-carboxamide
2-{4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
1-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
3-{[benzyl(methyl)amino]methyl}-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}(methyl)[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amine
1-[1-(1-{[1-(2-fluorophenyl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol