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N-(1H-imidazol-2-ylmethyl)-N-methyl-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(phenoxymethyl)-1-[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
3-[1-(2,5-dimethoxybenzenesulfonyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
ethyl 1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-2-carboxylate
3-(1-{2-[4-(methylsulfanyl)phenyl]acetyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
(3R,9aR)-8-[(3-fluoro-4-methylphenyl)methyl]-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-({2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
4-(4-fluorophenoxy)-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
3-methyl-N-{2-[1-(3,3,3-trifluoropropyl)piperidin-3-yl]ethyl}but-2-enamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(2,3-dimethoxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-{[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]sulfonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-{6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
N-benzyl-N-(1,3-thiazol-2-ylmethyl)oxane-2-carboxamide
2-methoxy-4-{4-[(3-methylphenyl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
1-(2-methoxyphenyl)-4-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]piperazine
1,3-dimethyl-5-{2-oxo-2-[3-(pyridin-2-yl)azetidin-1-yl]ethyl}imidazolidine-2,4-dione
1-({5-[1-(3,4-dimethylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)-4-methylpiperazine
4-cyclobutyl-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-6-methylpyrimidin-2-amine
{3-ethyl-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]piperidin-3-yl}methanol
9-[(2E)-3-phenylprop-2-en-1-yl]-3,9-diazaspiro[5.6]dodecane
2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}hexan-1-ol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-3-(1-methyl-1H-pyrazol-4-yl)propanamide
1-{4-[4-(4-phenylpiperazin-1-yl)piperidin-1-yl]benzoyl}piperidin-3-ol
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(1-methylcyclopentanecarbonyl)piperidin-4-ol
N-cyclopropyl-3-{5-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
4-(4-{[3-(1H-1,2,3-benzotriazol-1-yl)propyl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
4-[2-(furan-2-yl)-7-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperazine-1-carboxamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-(propan-2-yl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1-(2-methylphenyl)piperazin-2-one
(2R,3S,6R)-3-phenyl-5-(9H-purin-6-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methylpyrimidin-2-amine
N-(1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
methyl({[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl})[2-(morpholin-4-yl)ethyl]amine
[2-methoxy-5-(4-phenyl-1H-imidazol-1-yl)phenyl]methanol
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-4-(1H-1,2,4-triazol-3-yl)benzamide
1-(3-cyano-4-methylphenyl)-3-[2-(dimethylamino)ethyl]-3-[(5-methylthiophen-2-yl)methyl]urea
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(5-methyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-methyl-1-[1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidin-4-yl]butan-1-ol
8-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-methoxy-N-[(4-methoxyphenyl)methyl]-N-propylpyridine-4-carboxamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
2-(morpholin-4-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
7,7-dimethyl-2-{2-[methyl(phenyl)amino]ethyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
7-(cyclopropylmethyl)-2-(5,6-dimethylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-(4-phenyl-1,4-diazepane-1-carbonyl)-1-(propan-2-yl)pyrrolidin-2-one
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-(methylsulfanyl)pyridine-3-carboxamide
N-{2-oxo-4-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,3,4-tetrahydroquinolin-7-yl}acetamide
2-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
N-[3-(3-ethylphenoxy)propyl]-5-(methoxymethyl)-N-methylfuran-2-carboxamide