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2-methyl-7-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)-2,7-diazaspiro[4.4]nonane
N-[2-(3-chlorophenyl)ethyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-benzyl-4-acetamido-N-(3-hydroxy-2-methylpropyl)benzamide
1'-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
8-fluoro-2-[({5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}amino)methyl]quinolin-4-ol
4-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-6-(4-methyl-1H-pyrazol-1-yl)pyrimidine
5-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-N,N-dimethylpyridin-2-amine
3-(2-methoxyphenyl)-1-methyl-3-{2-[3-(2-methylphenyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
6-(3-hydroxyphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
1-[(4aR,8aR)-7-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
2-[(1-methylpiperidin-3-yl)methyl]-1,2-dihydroisoquinolin-1-one
2-(butylsulfanyl)-6-[3-(methanesulfonylmethyl)piperidin-1-yl]pyrimidin-4-amine
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-4-hydroxy-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidine-4-carboxamide
[(3R,4R)-1-(5-ethylthiophene-2-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
5-methyl-1-{2-[2-methyl-4-(2-methylphenyl)-5-oxopiperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-(3-chlorophenyl)-N,N-dimethyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(2,6-difluoro-3-methoxyphenyl)methyl]acetamide
3-({[2-(azepan-1-yl)ethyl](ethyl)amino}methyl)phenol
4-[(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]-5-(hydroxymethyl)-2-methylpyridin-3-ol
N-(adamantan-2-yl)-3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
(3R,4S)-1-(benzenesulfonyl)-4-cyclopropylpyrrolidin-3-amine
1-methyl-4-(1-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)piperazine
(3S,4R)-3-methoxy-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-4-amine
(1R,7S)-6-(2,3-dihydro-1H-isoindole-2-carbonyl)-3-[(3-methoxyphenyl)methyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
(2S)-2-[({2-[(2-chloroprop-2-en-1-yl)oxy]-6,7-dimethoxyquinolin-3-yl}methyl)amino]-4-methylpentanamide
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-[2-(propylsulfanyl)phenyl]urea
4-(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)pyrimidine
2-[(2-amino-6-{methyl[(1-phenyl-1H-pyrazol-4-yl)methyl]amino}pyrimidin-4-yl)amino]ethan-1-ol
methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})(1,3-thiazol-4-ylmethyl)amine
2-{9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carbonyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
5-{1-[(3,4,5-trimethoxyphenyl)methyl]-1H-imidazol-2-yl}pyrimidin-2-amine
3-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{3-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]piperidin-1-yl}pyrimidine
3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-8-(pyridin-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(azocan-1-yl)-3-[2-methoxy-4-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]propan-2-ol
(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-7-{[(3-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-(2-fluorophenoxy)-1-(3-methylfuran-2-carbonyl)piperidine-4-carboxylic acid
3-[(4-fluorophenyl)methyl]-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1,2-oxazole-5-carboxamide
4-{2-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}morpholine
7-(4,6-dimethylpyridine-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
5-({[6-(methoxymethyl)pyrimidin-4-yl]amino}methyl)-N-methylfuran-2-carboxamide
5-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}-4-propylpyrimidine
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-(pyrrolidin-1-yl)propanamide
9-[2-(4-methoxyphenoxy)acetyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
6-(azepan-1-yl)-N-[3-(1H-pyrazol-1-yl)propyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-{[6-oxo-2-(phenoxymethyl)-1,6-dihydropyrimidin-4-yl]methyl}acetamide
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-(2,5-dioxoimidazolidin-4-yl)acetamide
(2S)-2-amino-N-butyl-N-(furan-2-ylmethyl)-3-phenylpropanamide