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N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{[(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(3-methylphenoxy)piperidine
N-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-N-[(3-methylthiophen-2-yl)methyl]cyclopropanamine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
methyl 4-({[5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-yl]amino}methyl)benzoate
(3aR,6aS)-5-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
8-(2,1,3-benzoxadiazol-4-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-3-ol
1-[(1R,5R)-6-[(5-chlorothiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
(1R,5R)-6-(1H-imidazol-4-ylmethyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-chloro-5-[1-cyclohexyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
(1S,5R)-3-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-6-fluoroquinoline
(2S,4R)-1-(1H-imidazol-4-ylmethyl)-N-methyl-4-[2-(pyridin-2-ylsulfanyl)acetamido]pyrrolidine-2-carboxamide
(2R,3R)-1'-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[3-(2-methoxyphenyl)propyl]-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
2-{1-[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-2-yl}-1,3-thiazole
4-methoxy-N-{[1-(oxan-4-yl)piperidin-3-yl]methyl}benzene-1-sulfonamide
1-[2-(4-fluorophenyl)ethyl]-4-[(oxan-4-yl)amino]pyrrolidin-2-one
1-(cyclohexylmethyl)-6,7-dimethoxy-3-{[(pyridin-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
9-(2-methylpyrimidine-5-carbonyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[4-(2-hydroxyethyl)phenyl]-2-{4-[2-(1H-imidazol-1-yl)acetyl]morpholin-3-yl}acetamide
(3S,4R)-1-{2-[cyclopentyl(methyl)amino]acetyl}-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
1-[(2,4-dimethylphenyl)methyl]-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
2-(4-{4-[(ethylcarbamoyl)amino]-3-methoxyphenyl}phenyl)-N,N-dimethylacetamide
9-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-[4-(2,2-dimethylpropanamido)-3-methylphenyl]-1H-pyrazole-3-carboxamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-1-(pyrimidin-2-yl)piperidin-4-amine
2-{1-[(2-ethoxyphenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-phenoxypropan-1-one
2-cyclopropyl-9-[2-(2-ethylphenoxy)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-3-phenyl-N-(quinolin-5-ylmethyl)-1,2,4-oxadiazol-5-amine
4-{[1-(methoxymethyl)-1H-imidazol-2-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{4-[(2,3-difluorophenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
5-[4-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
2-[(3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)methyl]phenol
7-[(2-fluorophenyl)methyl]-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-[2-(methylsulfanyl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
5-{[2-(4-fluorophenyl)piperidin-1-yl]methyl}-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
6-cyclopentyl-2-methoxy-3-({[6-(methoxymethyl)pyrimidin-4-yl]amino}methyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(3aR,6aR)-2-acetyl-5-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-methyl-2-{1-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-1H-indole
3-[(dimethylamino)methyl]-1-(1H-indole-7-carbonyl)pyrrolidin-3-ol
4-(2-methoxyphenoxy)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
N,N-dimethyl-2-[4-(2-methyl-4-phenylpyridine-3-carbonyl)morpholin-3-yl]acetamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-propylacetamide