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1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(4-phenoxybenzoyl)piperidine
methyl 4-{[(3S,4S)-3-hydroxy-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-1-yl]methyl}benzoate
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
N-[cyclopropyl(pyridin-2-yl)methyl]-N,2,3,6-tetramethylquinoline-4-carboxamide
3-[(dimethylamino)methyl]-N-(5-fluoro-2-methoxyphenyl)-3-(hydroxymethyl)piperidine-1-carboxamide
N-{3-[(2R)-2-amino-3-methylbutanamido]phenyl}-2-methoxybenzamide
1-[2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(benzylsulfamoyl)-N-(furan-2-ylmethyl)piperidine-4-carboxamide
4-{2-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}-6-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-cyclopropyl-3-{5-[(2R)-oxolane-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-({[4-(1-methyl-1H-pyrazol-4-yl)phenyl]methyl}amino)propan-1-ol
{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}({[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl})amine
methyl 4-{[(2S)-2-carbamoylpyrrolidine-1-carbonyl]amino}benzoate
9-[(2S,3S)-2-amino-3-methylpentanoyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
5-chloro-2-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidine-1-carbonyl]phenol
N-[3-(1H-indol-1-yl)propyl]-5-methyl-1,3-oxazole-4-carboxamide
(1R,5R)-6-(cyclopropylmethyl)-3-[2-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
2-{[2-(N-methylmethanesulfonamido)ethyl]amino}-N-[1-(4-methylphenyl)ethyl]acetamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)amine
methyl 3-[({[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}carbamoyl)amino]benzoate
4-(2H-1,3-benzodioxol-5-yloxy)-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
1-(2-{4-[(4-phenylphenyl)methyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-[(4aS,8aR)-decahydroisoquinolin-2-ylmethyl]-N-(1,4-dimethyl-1H-pyrazol-5-yl)benzamide
(4aS,8aR)-1-(4-hydroxybutyl)-6-[2-(pyridin-4-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
methyl 6-(2,3-difluorobenzoyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[3-(furan-2-yl)-5-{[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]methyl}-1H-1,2,4-triazol-1-yl]butan-2-ol
2-(2,5-dioxoimidazolidin-1-yl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[2-(1H-indol-1-yl)ethyl]-N-methylpyrimidin-2-amine
N-[(3R,4R)-3-hydroxy-1-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl]pyrazine-2-carboxamide
3-(1H-pyrazol-5-yl)-1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperidine
5-acetyl-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(1-cyclopentyl-1H-pyrazol-5-yl)-2-{4-[6-methyl-2-(methylamino)pyrimidin-4-yl]-1H-pyrazol-1-yl}acetamide
N-[1-(3-methylphenyl)piperidin-4-yl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
N'-methyl-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-N'-phenylethanediamide
3-ethyl-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-4H-1,2,4-triazole
1-{2-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidin-4-yl}piperidin-3-ol
4-[1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]pyridine
[4-fluoro-7-(3-methoxypyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
2-(2-chlorophenyl)-2-hydroxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
(2S,4S)-4-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-amido}-N-ethyl-1-methylpyrrolidine-2-carboxamide
{4-[(4-methoxyphenyl)methyl]-1-(quinoline-8-sulfonyl)piperidin-4-yl}methanol
4-{3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}phenol
2-(3-fluorophenoxymethyl)-N-[1-(2-methylpropanoyl)piperidin-4-yl]-1,3-oxazole-4-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-{4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}ethan-1-one
4-{3-[2-(3-hydroxypropyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
1-tert-butyl-N-[2-(2-methoxynaphthalen-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
(3S,9aR)-8-(4-chlorobenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-chloro-N,2-dimethyl-N-{2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}benzene-1-sulfonamide
3-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one