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2-[4-(4-benzyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-4-carboxamide
1-(1H-imidazol-2-ylmethyl)-N-[3-(3-methylphenyl)phenyl]pyrrolidine-2-carboxamide
[(2-fluorophenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]pyrrolidine-1-sulfonamide
1-[(3,4-difluorophenyl)methyl]-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-(1,3-benzothiazol-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
5-methyl-N-(prop-2-en-1-yl)-6-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}thieno[2,3-d]pyrimidin-4-amine
(3R,9aR)-8-(2-methoxybenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-ethyl-2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
2-{2-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-6-methylpyridine
(3aR,5R,6S,7aS)-2-{[5-chloro-3-methoxy-2-(propan-2-yloxy)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
N-(3-phenylprop-2-yn-1-yl)-N-propylpiperidine-4-carboxamide
4-({[2-(pyrrolidin-1-yl)-6-(trifluoromethyl)pyrimidin-4-yl]amino}methyl)azepan-4-ol
(3aR,6aS)-5-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[4-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
5-{[(6-phenylpyridazin-3-yl)amino]methyl}pyrrolidin-2-one
5-{[1-(1H-1,3-benzodiazol-2-yl)ethyl]carbamoyl}-1H-imidazole-4-carboxylic acid
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(4-methoxyphenyl)methyl]-N-methyl-N-(quinolin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
methyl 3-{[(1,3-dimethyl-1H-pyrazol-5-yl)formamido]methyl}-5-[(2E)-3-(3-fluorophenyl)prop-2-enamido]benzoate
2-(4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
N,3-dimethyl-1-propyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
N-(2,2-diphenylpropyl)-4-hydroxy-1-methylpiperidine-4-carboxamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
3-methyl-1-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-1,2-dihydroquinoxalin-2-one
4-(1-ethyl-1H-imidazol-2-yl)-1-[4-(5-methylfuran-2-yl)benzoyl]piperidine
ethyl 4-[(4-chlorophenyl)methyl]-1-[3-(1-methylcyclopropyl)propanoyl]piperidine-4-carboxylate
1-{1-[2-(dimethylamino)acetyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-[(4-sulfamoylpiperazin-1-yl)methyl]benzoic acid
5-[({2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)methyl]-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-4-carbonitrile
1-[(4-fluorophenyl)methyl]-4-(3-propyl-1H-pyrazole-4-carbonyl)-1,4-diazepane
3-[(3R,4S)-4-(morpholin-4-yl)-1-[(5-phenylthiophen-2-yl)methyl]piperidin-3-yl]propan-1-ol
[(2S,6S)-4-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
2-[4-(dimethylamino)azepan-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(4aR,8aR)-2-cyclopentanecarbonyl-7-(pyrimidin-2-ylmethyl)-decahydro-2,7-naphthyridin-4a-ol
N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-[4-(3-methylphenyl)phenyl]-1-[3-(pyridin-4-yl)propanoyl]piperidine-4-carboxamide
1-(cyclopropylmethyl)-4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
N-[3-(3-benzyl-1H-1,2,4-triazol-5-yl)-5-methylthiophen-2-yl]-2,2-dimethylpropanamide
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}butan-1-one
1-{2-[(cyclohex-3-en-1-ylmethyl)amino]ethyl}-N-(thiophen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
N-[2-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)propyl]-2H-1,3-benzodioxole-5-carboxamide
methyl (2S,4S,5R)-5-(2,3-difluorophenyl)-1-methyl-4-{[(3-methylpyridin-2-yl)methyl]carbamoyl}pyrrolidine-2-carboxylate
N-(2-ethylphenyl)-3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carboxamide
3-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-7-methoxy-1-methyl-1,2-dihydroquinolin-2-one