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N-(6-chloro-2-methylpyridin-3-yl)-4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
N-butyl-N-[(5-methylthiophen-2-yl)methyl]-3-(6-oxo-1,6-dihydropyridazin-3-yl)propanamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methoxyhexan-1-one
(3S,9aR)-3-[(2S)-butan-2-yl]-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2S,4R)-1-[(3-chlorophenyl)methyl]-N,N-diethyl-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
7-[(4-fluorophenyl)methyl]-2-(thian-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(5-methylfuran-2-yl)ethyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(3-methyl-1,2-oxazol-5-yl)-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
(2S,4R)-4-amino-N-methyl-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide
(1R,3S)-1-hydroxy-3-methoxy-N-[2-(propan-2-yl)phenyl]-7-azaspiro[3.5]nonane-7-carboxamide
(4aR,7aS)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]-1-methylurea
4-(hydroxymethyl)-1-(2,3,4-trimethoxybenzoyl)piperidin-4-ol
2-{1-[(5-methylfuran-2-yl)methyl]-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
(1R,5R)-6-(2-methoxyethyl)-3-(5-propyl-1,3,4-thiadiazol-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(3aS,6aR)-5-(3-hydroxybenzoyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}furan-2-carboxamide
1-[(4-chlorophenyl)methyl]-N-[2-(2-methylphenyl)ethyl]-6-oxopiperidine-3-carboxamide
4-benzyl-3-butyl-1-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-cyclohexyl-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]pyrimidin-2-amine
1-(furan-2-ylmethyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
4-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butanamide
2-cyclopentyl-1-[3-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
N-(3,3-diphenylpropyl)-6-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-6-azaspiro[2.5]octane-1-carboxamide
N,N-dimethyl-2-(pyridin-2-yl)-7-[(2R)-pyrrolidine-2-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl[(2E)-3-phenylprop-2-en-1-yl]{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
1-(3-methoxybenzoyl)-4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperazine
N-{2-[1-(2-oxoazepan-3-yl)-1H-imidazol-2-yl]quinolin-6-yl}acetamide
(3S,4R)-1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(2R,6R)-4-[(4-methylpiperidin-1-yl)sulfonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-6-carboxylic acid
4-chloro-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
5-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
4-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]benzonitrile
N-cyclopentyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)ethane-1-sulfonamide
(1,4-dioxan-2-ylmethyl)(methyl){[2-(methylsulfanyl)phenyl]methyl}amine
N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1-[3-(1H-pyrazol-5-yl)phenyl]piperidin-4-amine
3-[(3S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-methylpropanamide
4-(4-chlorophenoxy)-N-[1-(pyridin-2-yl)propyl]piperidine-4-carboxamide
2-{3,5-dimethyl-4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1H-pyrazol-1-yl}acetic acid
3-{1,4-diazabicyclo[3.2.2]nonan-4-ylmethyl}-7-methyl-1,2-dihydroquinolin-2-one
1-[2-(benzyloxy)phenyl]-3-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-methylurea
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(cyclopentylmethyl)-1-(3-methoxypropyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
6-(2-chlorophenyl)-2-{4-[(3-oxopiperazin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N,N-dimethyl-5-({methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amino}methyl)pyridin-2-amine
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide