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1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butane-1,2-dione
(3S,4R)-4-(3-fluorophenyl)-1-[4-(4-methylphenyl)-4-oxobutyl]pyrrolidine-3-carboxylic acid
(4aS,7aR)-1-[(4-ethylphenyl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-ethyl-3-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
4-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2-methylphenol
N2-cyclopropyl-N4-[2-(1H-1,2,3-triazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
6-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
N-cyclopropyl-2-fluoro-N-[(2E)-3-phenylprop-2-en-1-yl]-5-sulfamoylbenzamide
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
methyl[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl][2-(pyridin-4-yl)ethyl]amine
(4aS,7aR)-1-[(2-chlorophenyl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-{4-[(4,4-dimethylpiperidin-1-yl)methyl]phenoxy}ethyl)-4-ethylpiperazine
1-(2-{[4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethyl)piperidin-2-one
2-(4-{[4-(2-methoxyphenyl)piperidin-1-yl]methyl}phenoxy)propanoic acid
4-(3-hydroxy-3-methylbutyl)-N-[(4-hydroxyphenyl)methyl]benzamide
({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]amine
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1H-1,2,3-benzotriazole-5-carboxamide
N5-[(2-chlorophenyl)methyl]-1-cyclopentyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-(3,5-dichlorophenyl)-6-methylpyridazine
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
2-[2-(4,4-difluoropiperidin-1-yl)-2-oxoethyl]-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
7-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
N-butyl-3-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(methylsulfanyl)phenyl]urea
3-(2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-oxoethyl)-5,5-dimethylimidazolidine-2,4-dione
N'1-{2-methyl-3-[(1,3-thiazol-2-yl)carbamoyl]phenyl}cyclopropane-1,1-dicarboxamide
3-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-(4-methoxyphenyl)-3-methyl-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-one
2,3,6-trimethyl-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)quinoline-4-carboxamide
methyl (2S)-2-{[1-(4-cyclopentaneamidophenyl)piperidin-4-yl]amino}-2-phenylacetate
2-{1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}pyridine
methyl 5-[(3-hydroxy-3-methylbutan-2-yl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-{2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-methyl-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
2-{6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[4-(piperidin-1-ylmethyl)phenyl]formamido}acetic acid
1-[(1-{6-[(thiolan-3-yl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-(2-hydroxyphenyl)ethan-1-one
3-methyl-N-{1-[1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-(3-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-(1-methylpiperidin-2-yl)propan-1-one
2-ethoxy-1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-methyl-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(propan-2-yl)acetamide
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide