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(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)(pyridin-4-ylmethyl)amine
1-methyl-3-(propan-2-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
1-methyl-4-{[5-(4-methyl-1,3-thiazol-5-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]methyl}piperidine
1-(1-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1,2,3,6-tetrahydropyridin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-(azepane-1-carbonyl)-N-methyl-1-(prop-2-en-1-yl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(5-methyl-1,2,4-oxadiazol-3-yl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-1-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetamide
1-[(2-chloro-4-fluorophenyl)methyl]-3-(3-methoxyphenoxy)azetidine
(4aR,8aR)-2-[(2-butyl-1H-imidazol-4-yl)methyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[1'-(furan-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
6-fluoro-2-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)quinolin-4-ol
5-(2-chloro-4-fluorophenoxymethyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
methyl 1-{5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}aziridine-2-carboxylate
2-amino-4-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
4-[4-(1,3-thiazol-4-yl)phenyl]-4H-1,2,4-triazole
N-cyclobutyl-3-{[4-(1H-pyrazol-1-yl)butan-2-yl]sulfamoyl}benzamide
6-{[(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amino]methyl}naphthalen-2-ol
3-{2-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-methoxy-N-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2-phenylacetamide
(3S,4S)-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
4-tert-butyl-2-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)phenol
N-[(1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
N-(1-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
2-tert-butyl-6-(oxane-2-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2,6-dimethoxypyrimidine-4-carboxamide
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine
1-[2-(3-methoxypyrrolidin-1-yl)-2-oxoethyl]-3-methyl-1,2-dihydroquinoxalin-2-one
3-butyl-1-methyl-4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperazin-2-one
1-[2-(4-methylpiperazin-1-yl)ethyl]-3-(2-phenyl-1-benzofuran-5-yl)urea
1-{1-ethyl-5-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-phenylpiperazine
7-cyclopentanecarbonyl-2-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2,7-diazaspiro[4.5]decane
2-cyclopropyl-9-(4-methylbenzoyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
(3S,4S)-1-(benzenesulfonyl)-4-[(1-benzothiophen-2-ylmethyl)(methyl)amino]pyrrolidin-3-ol
4-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4-oxobutanamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]naphthalene-2-sulfonamide
N-[(2-ethoxyphenyl)methyl]-N-ethyl-2-methyl-3-(1H-pyrazol-1-yl)propanamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)(thiophen-2-ylmethyl)amine
4-({4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzonitrile
4-chloro-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidine
4-methylphenyl (7S,9aR)-7-[(4-chlorophenyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-[(2S)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
1-(2-aminoethyl)-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-[2-(2-ethylphenoxy)ethyl]-N-methyl-2-(2-oxopiperidin-1-yl)acetamide
1-[(2-chlorophenyl)methyl]-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
3-({4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)-7-methyl-1,2-dihydroquinolin-2-one
N,6-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-2-oxo-1,2-dihydropyridine-4-carboxamide