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N-(2,3-dihydro-1H-inden-1-yl)-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
1-{[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]methyl}pyrrolidin-2-one
2-ethyl-9-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(piperidin-3-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]benzamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(3S,4R)-1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
methyl({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl})[1-(pyridin-3-yl)ethyl]amine
N-{1-[1-(2-hydroxyethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
4-methyl-2-[1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
2-[4-methyl-6-({4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amino)pyrimidin-2-yl]phenol
4-{[3-(3-carboxyphenyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
N,N-dimethyl-1-({2-[3-(4-methylpiperazin-1-yl)propoxy]phenyl}methyl)piperidin-3-amine
N,N-dimethyl-1-[(1-methylazepan-2-yl)methyl]piperidin-3-amine
5-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
7-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{[(1,3-thiazol-2-yl)carbamoyl]methyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-(3-{2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethoxy}phenyl)propanamide
N-[4-(methylamino)butyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
6-{3-methyl-3,9-diazaspiro[5.6]dodecane-9-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
3-[2-(2,4-difluorophenyl)ethyl]-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
2-methyl-2-(morpholin-4-yl)-1-[3-(2-phenylacetyl)piperidin-1-yl]propan-1-one
(3S,4S)-3-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-4-hydroxy-1λ6-thiolane-1,1-dione
3-({3-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}methyl)pyridin-2-amine
1-{2-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)phenoxy]ethyl}-1H-imidazole
2-(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
1-[2-(4-methoxyphenyl)ethyl]-8-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-hydroxy-1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}piperidine-4-carboxylic acid
(2E)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-4-methylpent-2-enamide
3-{[(3-hydroxy-2,2-dimethylpropyl)(methyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-{2-[(dimethylamino)methyl]-4-(pyrimidin-2-yl)phenoxy}-N-[2-(3-fluorophenyl)ethyl]acetamide
N'-(2-chlorophenyl)-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]ethanediamide
4-phenyl-2-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]pyrimidine
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyridin-2-amine
9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(4-methylphenoxy)ethan-1-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
3-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-3-phenyl-N-(pyridin-4-ylmethyl)butanamide
5-oxo-1-(pyridin-3-ylmethyl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyrrolidine-3-carboxamide
3-(1-methyl-1H-imidazol-4-yl)-5-[3-(1H-pyrazol-4-yl)phenyl]-1,2,4-oxadiazole
9-{1-[(4-methylphenyl)amino]cyclohexanecarbonyl}-1,4,9-triazaspiro[5.5]undecan-5-one
N-cyclopropyl-1-[(1s,4s)-4-(2,4-difluorobenzenesulfonamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
(2S,4R)-N-ethyl-4-[2-(1H-imidazol-1-yl)acetamido]-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
3-cyclopropyl-1-(4-methoxyphenyl)-5-(1H-pyrazol-1-ylmethyl)-1H-1,2,4-triazole
1-[5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(propylsulfanyl)ethan-1-one
(1S,5R)-N-(4-acetylphenyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-[6-hydroxy-4-(1H-imidazol-2-ylmethyl)-1,4-diazepan-1-yl]-2-(2-methylphenyl)ethan-1-one
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(1H-1,2,4-triazol-3-yl)benzamide
1-(4-fluorophenyl)-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]cyclopropane-1-carboxamide