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N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-2-methanesulfonyl-N-methylacetamide
3-(3-fluoro-4-methoxybenzoyl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine
1-ethyl-N,N-dimethyl-3-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazol-5-amine
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidine
N-[2-(3-fluorophenyl)ethyl]-2,2-dimethyloxane-4-carboxamide
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
2-fluoro-6-[4-(propan-2-yloxy)phenyl]benzamide
1-[(2-methylphenyl)methyl]-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
2-(azepan-1-yl)-2-[4-(2-methoxyethoxy)phenyl]acetic acid
2,3-dimethyl-7-[3-(morpholin-4-yl)propanoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-(3-chloro-2,6-difluorophenyl)-1-(3-methoxypropyl)-1H-imidazole
1-[cyclohexyl(methyl)amino]-3-(3-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)propan-2-ol
3-{5-[(4-fluoro-3-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
ethyl 4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazine-1-carboxylate
3-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)-1-ethyl-1-(oxan-4-ylmethyl)urea
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-[(4-methylpiperidin-1-yl)methyl]piperidin-2-one
N-benzyl-6-(3-phenylprop-2-ynoyl)-6-azaspiro[2.5]octane-1-carboxamide
1-(4-methyl-1H-pyrrole-2-carbonyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
1-[3-(2-oxopyrrolidin-1-yl)propyl]-3-[1-(1-phenylethyl)-1H-pyrazol-5-yl]urea
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(4-methyl-2-oxopyrrolidin-1-yl)acetamide
(2S,4R)-1-[(2,4-dimethylphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
4-{2-[2-(dimethyl-1,2-oxazol-4-yl)-1H-imidazol-1-yl]-1-(pyridin-2-yl)ethyl}morpholine
(2S,4R)-N-methyl-4-[4-(2-{[(4-methylphenyl)carbamoyl]amino}propan-2-yl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
5-fluoro-2-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-2-yl}-1H-1,3-benzodiazole
5-methoxy-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
4-{[2-(4-methoxyphenyl)ethyl]amino}-N,5-dimethyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
(2S,4R)-N-methyl-1-(oxan-4-yl)-4-[2-(phenylsulfanyl)acetamido]pyrrolidine-2-carboxamide
3-[3-(4-fluorophenyl)oxolan-3-yl]-5-(thiophen-3-yl)-1,2,4-oxadiazole
1-(4-methyl-3-phenylpiperazin-1-yl)-3-(pyridin-3-yl)propan-1-one
2-(dimethylamino)-2-(4-fluorophenyl)-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}acetamide
1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2-amino-4-(4-hydroxy-3,5-dimethoxyphenyl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
(2R,6S)-2,6-dimethyl-N-(2-methyl-1-benzofuran-7-yl)morpholine-4-carboxamide
(4aR,7aS)-1-{2-[4-(aminomethyl)piperidin-1-yl]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-2-[({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]acetamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{[1-(2-amino-1,3-benzothiazole-5-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
2-chloro-6-ethoxy-4-{[(1H-imidazol-2-ylmethyl)amino]methyl}phenyl acetate
N-cyclohexyl-N-methyl-4-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-4-oxobutanamide
methyl 2-({2-[(3-methoxyphenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}amino)acetate
4-[2-(cyclopropylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-N,N-dimethylpiperazine-1-carboxamide
2-{4-[(5-methylfuran-2-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
6-methyl-5-{2-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[4-(diphenylmethyl)piperazin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-(1-methanesulfonylpyrrolidine-2-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
2-benzyl-4-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-3-methyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-{1-[(3,4-difluorophenyl)methyl]-4-(3-methyl-1H-pyrazole-5-carbonyl)piperazin-2-yl}ethan-1-ol
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]pyridine-2-carboxamide
(3R,5R)-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide