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6-methyl-5-(quinolin-8-yl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S)-N-[2-(2,5-dimethylphenoxy)ethyl]piperidine-2-carboxamide
3-{1-ethyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}-1-methyl-1,2-dihydroquinoxalin-2-one
3-[5-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1-benzyl-4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-amino-3-ethyl-N-[2-(pyridin-4-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(7-fluoro-4-methylquinolin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(2,5-dimethylphenyl)methyl]-2-(3-hydroxyadamantan-1-yl)acetamide
5-fluoro-2-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
(3S,4S)-3,4-bis(hydroxymethyl)-N-[2-(3-methylphenyl)-1,3-benzoxazol-6-yl]pyrrolidine-1-carboxamide
3-(3-hydroxyquinoxalin-2-yl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
4-(benzyloxy)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]butan-1-one
2-[4-(5-methylthiophene-3-carbonyl)piperazin-1-yl]-1,3-benzothiazole
9-(cyclopropylmethyl)-4-(3-hydroxy-2-methylbenzoyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-phenyl-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-ynamide
1-(2-{[2-(4-hydroxy-3-methoxyphenyl)ethyl]amino}pyrimidin-4-yl)piperidin-3-ol
(3E)-N-[3-(2-phenylacetamido)phenyl]hex-3-enamide
3-{[1-(azepane-1-sulfonyl)piperidin-4-yl]methyl}benzoic acid
6-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
N-[(2-ethoxyphenyl)methyl]-2-(methylsulfanyl)-6-oxo-N-(prop-2-en-1-yl)-1,6-dihydropyrimidine-5-carboxamide
1-(3-chlorophenyl)-4-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N-ethyl-5-phenyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
(4aS,7aR)-1-[(4-ethylphenyl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,7S)-3-(2-ethylbutyl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-methyl-4-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}imidazolidin-2-one
3-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-5-[(propan-2-yl)sulfamoyl]benzamide
{4-[(2-chlorophenyl)methyl]-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl}methanol
1-(2-chloroprop-2-en-1-yl)-7-methyl-3-({[3-(morpholin-4-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
7-(2-hydroxyethyl)-2-{[2-(trifluoromethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-1-benzothiophene-2-carboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-(1H-pyrazol-4-yl)propanamide
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]oxane-4-carboxamide
1-benzyl-N3-cyclohexyl-N3-methyl-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-3-ethynyl-N-(oxolan-2-ylmethyl)benzamide
2-(3-methyl-2,5-dioxoimidazolidin-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
(3R,5S)-1-benzyl-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[(2-methoxyphenyl)methyl]piperidine-3-carboxamide
N-[3-(4-fluorophenyl)phenyl]-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxamide
(3R,4S)-4-cyclopropyl-1-[1-(3,4-dimethoxyphenyl)cyclopentanecarbonyl]pyrrolidin-3-amine
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-3-ol
N-(4-{[(1-cycloheptyl-5-oxopyrrolidin-3-yl)amino]methyl}phenyl)acetamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(propan-2-yloxy)propyl]acetamide
2-(3-chloro-4-hydroxyphenyl)-N-methyl-N-[1-(pyridin-4-yl)ethyl]acetamide
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methylphenol
[(2S,6S)-4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
2-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
1-[(dimethylcarbamoyl)methyl]-N-[3-(3-methoxyphenyl)phenyl]piperidine-2-carboxamide
8-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-fluorophenyl)-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazole-4-carboxamide
2-(dimethylamino)-7-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]acetyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one