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4-[1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)piperidin-3-yl]benzoic acid
N-[4-(4-{[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
3-(azepan-1-yl)-1-[4-(2-methoxybenzoyl)piperazin-1-yl]propan-1-one
2-[1-(3-methyl-1H-pyrazole-5-carbonyl)azetidin-3-yl]pyridine
N,2-dimethyl-3-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
6-ethyl-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}pyrimidin-4-amine
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-[(8-methylquinolin-5-yl)methyl]pyrrolidin-3-yl]methanol
6-tert-butyl-1-methyl-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,4S)-4-cyclopropyl-1-[3-(thiophen-3-yl)propanoyl]pyrrolidine-3-carboxylic acid
1-[(3-chlorophenyl)methyl]-4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazine
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N,N,4-trimethylpyrimidin-2-amine
N-[2-(methylamino)ethyl]-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[(dimethylamino)methyl]piperidin-4-ol
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3,4-dimethoxybenzamide
2-{3-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
1-[3-(pyridin-3-yl)azetidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-(2,3-dihydro-1H-inden-1-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}acetamide
4-({2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)-1,5-dimethyl-1H-pyrrole-2-carbonitrile
2-[5-(4-acetylphenoxymethyl)-1-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]acetamide
4-[(cyclopropylmethyl)amino]-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
2-[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]-N-[2-methyl-6-(propan-2-yl)phenyl]acetamide
6-{[(2-hydroxypyridin-3-yl)methyl]amino}-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
N-(piperidin-4-ylmethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-({[2-(1H-1,3-benzodiazol-2-yl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
(4aS,8aR)-6-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
2-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4-(1H-1,2,3,4-tetrazol-1-yl)phenol
2-(2,3-dihydro-1H-isoindol-2-yl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
1-cyclopentyl-4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}pyrrolidin-2-one
2-{[2-(pyridin-2-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
6-fluoro-2-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}quinolin-4-ol
N-methyl-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(3-phenyl-1,2-oxazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-(1H-indol-2-ylmethyl)-2-[N-(3-methylphenyl)methanesulfonamido]acetamide
2-{5-[2-(1H-indol-3-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[5-(morpholin-4-yl)pentyl]thiolan-3-amine
2-(2-chlorophenyl)-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]acetamide
14-(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(3S,4R)-4-methyl-1-[1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carbonyl]-3-(2-methylpropyl)piperidin-4-ol
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
2-(1-{[1-(butane-1-sulfonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
1-{2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[1-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
3-[4-(dimethylamino)phenyl]-1-[(3S)-3-ethylmorpholin-4-yl]propan-1-one
1,5-dimethyl-4-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-[2-methoxy-4-({[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-amine
N3-(butan-2-yl)-1-cyclopentyl-4-oxo-N5-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-hydroxypropan-1-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-4-carboxamide
methyl 3-{[(3,5-dimethylphenyl)formamido]methyl}-5-(furan-2-amido)benzoate