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2-(2,6-difluorophenyl)-N-[(1-propylpiperidin-4-yl)methyl]acetamide
4-chlorophenyl (7S,9aR)-7-[(2S)-butan-2-yl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)-N-[(3-methoxyphenyl)methyl]propanamide
2-methoxy-N-[2-(pyridin-2-ylsulfanyl)ethyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-[3-(2,5-dimethylphenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
6-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
2-methyl-1-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}-1,4-diazepan-5-one
2-[4-(2,2-dimethoxyethyl)piperazin-1-yl]acetic acid
3-{[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl}-N-(pyridin-3-yl)benzamide
7-(2-methoxyethyl)-2-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-2,7-diazaspiro[4.5]decane
4-[4-(furan-2-yl)benzoyl]-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
1-cyclohexyl-5-(1-methyl-1H-pyrazol-4-yl)-1H-1,2,4-triazole
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]acetamide
1-(furan-2-carbonyl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
4-(1-benzyl-4-phenylpiperidine-4-carbonyl)morpholine
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)acetamide
2-(2-hydroxyethyl)-8-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
[(2-butoxy-3-methoxyphenyl)methyl][(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]amine
1-cyclopentyl-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]piperidine-3-carboxamide
1-[(5-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}thiophen-2-yl)methyl]piperidine
N-(3-methoxyphenyl)-5-(1-methyl-1H-pyrazol-4-yl)furan-2-carboxamide
2-(cyclopropylmethyl)-9-[(2-fluoro-5-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
4-[2-(3-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-2-methoxypyridine-3-carbonitrile
N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
7,7-dimethyl-2-(oxolan-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[(3S,4R)-1-benzyl-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-N-(4-methoxyphenyl)propanamide
methyl 2-{1-[(7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-3-oxopiperazin-2-yl}acetate
1-[1-(2,2-diphenylethyl)piperidin-3-yl]-4-phenylpiperazine
4-(dimethyl-1,3-thiazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-phenyl-4-[(2,3,4-trimethoxyphenyl)methyl]-1,4-diazepane
(1R,9S)-5-amino-3-(thiophen-3-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
3-methyl-5-{[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1,2-oxazole
2-methyl-N-[1-(pyrazin-2-yl)piperidin-4-yl]-1-benzofuran-5-carboxamide
5-(8-methoxyquinolin-5-yl)-N-methylthiophene-2-carboxamide
(3-{2-[1-(1H-1,2,3-benzotriazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
2-{2-[2-(3-methoxyphenoxy)ethyl]phenyl}-5-methyl-1,3,4-oxadiazole
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-2-methoxypyridine-4-carboxamide
3-{[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]methyl}-1,3-diazinane-2,4-dione
2-hydroxy-1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
(1S,5R)-6-methyl-3-[4-(trifluoromethyl)benzenesulfonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{[3,3-dimethyl-1-(pyridin-3-yl)butyl]amino}-N-(propan-2-yl)pyridine-2-carboxamide
1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxylic acid
3-[5-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
2-{methyl[(4-methyl-5-{1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amino}ethan-1-ol
1-(2-methylpyridin-4-yl)-4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-1,4-diazepane
3-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)propanamide
N-ethyl-5-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyrimidin-2-amine