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5-[(1-oxo-1,2-dihydroisoquinolin-2-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
1-ethyl-3-methyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1H-pyrazole-4-carboxamide
3-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N,N-dimethylaniline
[1-(1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-2-phenylethyl](methyl)(pyridin-4-ylmethyl)amine
(3aR,6aR)-2-(cyclobutylmethyl)-5-(pyridin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4,6-dimethylpyrimidin-2-yl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
1-(4-fluoro-3-methylbenzoyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-propylacetamide
N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
6-(3-methoxypyrazin-2-yl)-2-methyl-3,4-dihydroquinazolin-4-one
3-(3-methoxypropyl)-1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidine-3-carboxylic acid
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(2-methyl-1-benzofuran-7-carbonyl)piperidine
2-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-benzofuran-5-carboxamide
1-[1-(2-phenylethyl)piperidin-4-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
3-(1-methyl-1H-pyrazol-5-yl)-N-[(4-methylphenyl)(thiophen-2-yl)methyl]propanamide
5,6,7-trimethoxy-N,N-dimethyl-3-{[(thiophen-2-ylmethyl)amino]methyl}quinolin-2-amine
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
methyl 4-oxo-4-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)butanoate
N-(4-methoxy-2-methylphenyl)-3-[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]propanamide
9-{[4-(2-methylpropyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-(2,2-difluorocyclopropanecarbonyl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
1,3-dimethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(1R,5R)-6-[(2-ethoxyphenyl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(pyridin-3-ylmethyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine-2-carboxamide
4-(4-fluorophenyl)-1-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-ol
2-[3-(morpholin-4-ylmethyl)phenyl]-6-(phenoxymethyl)-3,4-dihydropyrimidin-4-one
methyl 4-methyl-3-({7-methyl-2,7-diazaspiro[4.4]nonane-2-carbonyl}amino)benzoate
N-methyl-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
5-cyclopropyl-N-(2-methoxyethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-(3-methoxyphenyl)-4-(pyrazin-2-yl)piperazin-2-one
4-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1,4-oxazepan-6-ol
methyl 4-[({1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidin-3-yl}formamido)methyl]benzoate
6-fluoro-N-methyl-N-(propan-2-yl)-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
(5S)-5-{[benzyl({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
N-benzyl-N-methyl-2-{[(pyridin-2-ylmethyl)amino]methyl}-2,3-dihydro-1H-inden-2-amine
(4aS,7aR)-1-(4-hydroxy-3-methylbenzoyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(3-ethylpiperazin-1-yl)-N-(pyridin-2-ylmethyl)pyridine-2-carboxamide
8-cyclopropanecarbonyl-2-(thiophen-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(2,3-dihydro-1H-inden-2-yl)-5-methoxyfuran-2-carboxamide
N,N-dimethyl-4-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]piperidine-1-carboxamide
6-fluoro-2-({[2-(1H-imidazol-4-yl)ethyl]amino}methyl)quinolin-4-ol
N-{[7-(3-chlorothiophene-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
1-[6-hydroxy-4-(3-hydroxypropyl)-1,4-diazepan-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
1-(3-methylfuran-2-carbonyl)-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-2-(4-methoxyphenyl)ethan-1-one
6-cyclopentyl-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine