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1-(4,4-difluoropiperidin-1-yl)-4-(1H-pyrazol-4-yl)butan-1-one
{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}({3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)methylamine
1-methanesulfonyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}piperidin-4-amine
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)oxane-4-carboxamide
(3S,4R)-1-(1H-imidazol-2-ylmethyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
2-{[2-(2-chloro-4-fluorophenyl)ethyl](propan-2-yl)amino}ethan-1-ol
4-[2-(3-chloro-4-fluorophenoxy)acetyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-ol
4-(2,2-dimethyloxane-4-carbonyl)-7-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
(3R,5S)-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}pyrrolidin-3-amine
(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
N-({5-[(2-phenoxyethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)pyridine-4-carboxamide
4-{4-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]phenyl}-4H-1,2,4-triazole
N,4-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,2,3-thiadiazole-5-carboxamide
(2R)-N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-cyclohexyl-2-hydroxyacetamide
1-ethyl-4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
3-(5-{1-[1-(furan-2-carbonyl)piperidin-3-yl]-1H-imidazol-2-yl}thiophen-3-yl)prop-2-yn-1-ol
(2S,4R)-4-amino-1-[2-amino-6-(2-methylpropyl)pyrimidine-4-carbonyl]-N-ethylpyrrolidine-2-carboxamide
4-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1λ6-thiane-1,1-dione
N-benzyl-2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazine-1-sulfonamide
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-(3,5-dimethylphenyl)propan-1-one
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[1-(hydroxymethyl)cyclopropanecarbonyl]pyrrolidine-3-carboxylic acid
1-[1-(3-tert-butyl-1,2,4-oxadiazol-5-yl)propyl]-2-ethyl-1H-1,3-benzodiazole
2-(dimethyl-1,3-thiazol-5-yl)-N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]acetamide
2-(3,4-dimethoxyphenyl)-5-fluoro-1-[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2,2-bis(prop-2-en-1-yl)-1-(2,3,4-trimethoxybenzoyl)piperidine
2-[3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]-1,3-thiazole-4-carboxamide
2-(2,4-dichlorophenoxy)-N-ethyl-N-(oxan-4-ylmethyl)acetamide
9-[2-(4-fluoro-3-methylphenyl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[5-(1-cyclopentanecarbonylpiperidin-4-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl]acetic acid
5-oxo-1-(pyridin-3-ylmethyl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)pyrrolidine-3-carboxamide
[(4-methoxyphenyl)methyl](methyl)({3-methyl-1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-4-yl}methyl)amine
N-[(5-methylpyrazin-2-yl)methyl]-5-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)pentanamide
N-cyclopentyl-4-{4-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]piperidin-1-yl}benzamide
methyl (2R)-2-{[2-(2-phenylethyl)-1,3-benzoxazol-5-yl]formamido}propanoate
9-[4-(5-methylfuran-2-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
(1R,5R)-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3-hydroxyquinoxalin-2-yl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}propanamide
5-({1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}carbamoyl)-2,1,3-benzoxadiazol-1-ium-1-olate
5-amino-3-[5-(1H-pyrazol-3-yl)furan-2-yl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
(5-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}furan-2-yl)methanol
1-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-2-[methyl(piperidin-4-yl)amino]ethan-1-one
4-ethyl-2-methyl-6-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
5-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-imidazol-2-yl}-N,N-dimethylpyridin-2-amine
1-{4-[3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]phenyl}-4-methylpiperazine
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
4-(1-benzofuran-5-carbonyl)-1-(4-methoxyphenyl)-2,2-dimethylpiperazine