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3-[(2-fluorophenyl)formamido]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]propanamide
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1-(9H-purin-6-yl)piperidin-4-amine
N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}-5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
N-(4-{2-[(methylcarbamoyl)methyl]-3-oxopiperazine-1-carbonyl}phenyl)pentanamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-4-chloro-1H-pyrazole-3-carboxamide
4-cyano-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1-methyl-N-(oxolan-2-ylmethyl)-1H-pyrrole-2-carboxamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(3-fluorophenyl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
1-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-2,3,4,9-tetrahydro-1H-carbazole
2-(1-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)-1,3-benzoxazole
6-[4-(5-methylpyridin-2-yl)-4-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
4-(thian-4-yl)-N-[4-(trifluoromethoxy)phenyl]piperazine-1-carboxamide
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-3-(thiophene-2-carbonyl)piperidine
4-ethyl-1-methyl-3-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl){[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
ethyl 2-[(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)amino]acetate
2-(2-methyl-1H-imidazol-1-yl)-1-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidin-1-yl}ethan-1-one
1-(4-methylphenyl)-4-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}piperazin-2-one
2-(1-{[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
N-[1-(1-cyclobutylpiperidin-4-yl)-2-(2-fluorophenyl)ethyl]-N-methylthiophene-3-carboxamide
N-(1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-yl)acetamide
(1H-imidazol-2-ylmethyl)(methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
2-(2-methoxyphenyl)-5-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidine
4-{[3-(4-fluorophenoxy)azetidin-1-yl]methyl}-1,4-dimethylpiperidine
1-{2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}azepan-2-one
2-(5-{[3-(pyridin-4-yl)azetidin-1-yl]methyl}furan-2-yl)benzonitrile
8-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
1-(2-methyl-1-benzofuran-7-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-methyl-4-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}-N-phenylaniline
N-(2-chlorophenyl)-4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
N-{4-fluoro-3-[({2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}carbamoyl)amino]phenyl}propanamide
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]cyclopent-3-ene-1-carboxamide
N-methyl-2-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-N-(propan-2-yl)acetamide
4-[({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-1-ethyl-N,N-dimethylpiperidin-4-amine
4-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-1,2-dimethylpiperazine
(1S,5R)-6-(2-methoxyethyl)-3-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(1-benzyl-1H-pyrazol-4-yl)-4-methylpyridin-2-amine
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]acetamide
(4aR,8aS)-1-[2-(3,4-difluorophenyl)acetyl]-N,N-dimethyl-decahydro-1,6-naphthyridine-6-sulfonamide
4-(5-methylpyridin-2-yl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-ol
3-amino-N-({1-[(2E)-2-ethylbut-2-en-1-yl]pyrrolidin-3-yl}methyl)benzamide
1-cyclooctyl-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
1-{3-[({5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)methyl]piperidin-1-yl}ethan-1-one
3-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1H-indole
3-(diphenylmethyl)-5-(oxolane-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-methyl-1H-pyrazole-4-carboxamide
2-amino-4-(4,5-dimethylfuran-2-yl)-6-propyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(furan-3-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
2-ethyl-N-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]pyrimidine-5-carboxamide
5-oxo-N-[2-(propane-2-sulfonyl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide