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3-(1-methyl-1H-imidazole-2-carbonyl)-1-(oxane-4-carbonyl)piperidine
1'-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]spiro[indene-1,4'-piperidine]
methyl 2-[2-(4-chlorophenyl)morpholin-4-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxylate
N-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
3-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-1-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
[3-(2-methoxyethyl)-1-(1H-1,2,3-triazole-5-carbonyl)piperidin-3-yl]methanol
7-(3-chlorophenyl)-9-methoxy-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[4-({4-[3-(prop-2-en-1-yloxy)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-ol
4-{[(3S,5R)-1-[(3,4-dimethoxyphenyl)methyl]-5-(pyrrolidine-1-carbonyl)piperidin-3-yl]methyl}morpholine
N-[3-(dimethylamino)-2,2-dimethylpropyl]-N'-(2-fluoro-5-methylphenyl)butanediamide
N-{3-[methyl(phenyl)amino]propyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
4-[(3,4-difluorophenyl)methyl]-9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-methyl-4-[(6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-yl)methyl]piperazine
3-[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]propanamide
(5S,9aS,9bS)-2-(3-methoxyphenyl)-5-(thiophen-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(4S)-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
5-(3-phenyl-1H-pyrazol-1-yl)pyridin-3-amine
5-(2-chloro-4-methoxyphenoxymethyl)-3-(pyrrolidine-1-carbonyl)-1H-pyrazole
1-cyclohexyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[2-(azocan-1-yl)-2-oxoethyl]-4-[(2,4-dimethoxyphenyl)methyl]piperazin-2-one
5-{[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]formamido}pentanoic acid
2-[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]-5-methyl-1H-1,3-benzodiazole
(1R,9S)-5-amino-3-(4-methanesulfonylphenyl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-{4-[3-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}acetamide
5-(morpholin-4-yl)-2-(4-phenoxybutyl)-2,3-dihydropyridazin-3-one
N,N-dimethyl-5-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}pyridin-2-amine
2-{3-[(3-chlorophenyl)methyl]-5-[(1,4-dimethylpiperazin-2-yl)methyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-(4-fluoro-2-methylphenyl)-3-[1-(thiophen-2-ylmethyl)piperidin-3-yl]propanamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
methyl 6-{[(butan-2-yl)(cyclopentyl)amino]methyl}pyridine-2-carboxylate
[2-(2-{1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)ethyl]dimethylamine
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-4-sulfamoylbutanamide
2-methyl-5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}phenol
2-(3-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}piperidin-1-yl)acetamide
3-[(2-methyl-1H-imidazol-1-yl)methyl]-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidine
N-[(4,6-dimethylpyridin-3-yl)methyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
4-[(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]benzonitrile
7-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]-2,4-dimethyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
4-{[7-(1-benzothiophen-3-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-ethyl-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}propan-1-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-methyl-5-(propan-2-yl)furan-3-carboxamide
N-methyl-2-(7-methyl-3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)-N-(thian-4-yl)acetamide
1-(4-methyl-1H-imidazole-5-carbonyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)[(2-phenyl-1,3-oxazol-4-yl)methyl]amine
2-ethyl-5-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
2-tert-butyl-6-(2-ethoxybenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-amino-4-(6-methylquinolin-5-yl)-6-(pyridin-3-yl)pyridine-3-carbonitrile
4-{3-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]propanamido}benzamide