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N-[(1-hydroxycyclohexyl)methyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
5-(2-chloro-4-fluorophenoxymethyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-ethyl-2-[3-(methoxymethyl)pyrrolidin-1-yl]pyridine-3-carboxamide
2-amino-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)-4-[2-(propan-2-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
5-fluoro-2-[1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
4-(pyridin-2-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]pyrimidin-2-amine
1-[6-hydroxy-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-1-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
N3-cyclooctyl-N5-[(5-methylfuran-2-yl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
2-(2-hydroxyethyl)-3-oxo-N-[(1R)-1-phenylethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-ethyl-5-[6-fluoro-4-(piperidine-1-carbonyl)quinolin-2-yl]pyrimidin-2-amine
2-{2-[(oxolan-2-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
N,N-diethyl-3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-(2,6-difluoro-4-methoxyphenyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-imidazole
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-(4-methylphenoxy)piperidine-4-carboxamide
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)pyrazine-2-carboxamide
5-[(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)carbamoyl]-1H-imidazole-4-carboxylic acid
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[2-(4-methylphenoxy)ethyl]-1,2-oxazole-3-carboxamide
2-(4-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
1-(1-propylpiperidin-4-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
2-[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-N,N-dimethylacetamide
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-cyclohexyl-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-amino-N-[2-(1-benzothiophen-2-yl)phenyl]acetamide
4-(1-{1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]piperidin-4-yl}ethyl)morpholine
(3aS,6aR)-5-(1-benzofuran-2-ylmethyl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(3aS,6aS)-2-ethyl-5-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
4-{1-[(4-methanesulfonylphenyl)methyl]pyrrolidin-2-yl}-3,5-dimethyl-1,2-oxazole
1-{7-[cyclohexyl(methoxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
N-[(1-ethylpyrrolidin-3-yl)methyl]-4-methoxy-N-methyl-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
4-(2-ethoxypyridine-3-carbonyl)-1-(2-methylphenyl)piperazin-2-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
2-ethyl-N-(2-phenoxyethyl)pyrimidine-5-carboxamide
2,7-dimethyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(1H-imidazol-2-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzamide
(1R,7S)-N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-({4-[3-(3-methylphenyl)piperidine-1-carbonyl]furan-2-yl}methyl)morpholine
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-[(4-methylphenyl)methyl]piperidine
3-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}benzonitrile
N-[(2,3-dichlorophenyl)methyl]-2-(1-methylpiperidin-2-yl)acetamide
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(1-benzothiophen-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-[(4-fluorophenyl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]piperidine
4-(1H-indazole-3-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
4-fluoro-3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzene-1-sulfonamide