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7-(2-methoxyethyl)-2-[2-(3-methylphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-phenyl-N-(1-phenylethyl)-1H-imidazole-4-carboxamide
(1S,5R)-N-(3-methoxyphenyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
4-[2-(5-acetylthiophen-3-yl)acetyl]-3-benzylpiperazin-2-one
7-fluoro-2-oxo-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1,2-dihydroquinoline-4-carboxamide
5-{[(2,3-dihydro-1H-inden-2-yl)(methyl)amino]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
N-[1-(1H-pyrazol-1-yl)propan-2-yl]-4-(pyridin-3-yl)pyrimidin-2-amine
4-[(1R,7S)-3-cycloheptyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carbonyl]-1λ6-thiomorpholine-1,1-dione
ethyl 4-oxo-5-phenoxy-1-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1,4-dihydropyridine-3-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(1,3-benzothiazol-2-yl)-N-(1-propyl-1H-pyrazol-5-yl)pyrrolidine-1-carboxamide
N,1,3-trimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-(ethylsulfanyl)-5-[1-(1,2-oxazol-3-ylmethyl)-4-phenyl-1H-imidazol-5-yl]pyrimidine
{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]amine
methyl 2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]pyridine-3-carboxylate
N-{[7-fluoro-5-(3-fluoro-4-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-3-yl)propanamide
methyl (2S,4R)-1-methyl-4-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)pyrrolidine-2-carboxylate
2-[methyl(1,2-oxazol-3-ylmethyl)amino]-2-[4-(2-methylpropanamido)phenyl]acetic acid
3-(4-hydroxyphenyl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1H-pyrazole-5-carboxamide
3-(4-methoxyphenyl)-N-methyl-3-phenyl-N-(pyridin-2-ylmethyl)propanamide
N-{2-[3-(morpholin-4-ylmethyl)phenoxy]propyl}furan-2-carboxamide
3-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidine-1-carbonyl}-6-(propan-2-yl)-1,2-dihydropyridin-2-one
(2S)-2-({2-methyl-3-[(pyridin-2-ylmethyl)amino]phenyl}formamido)-3-phenylpropanamide
6-ethoxy-3-{[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-(2-methoxyphenyl)-3-[1-(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
1-[1-(3-aminopropyl)-1H-1,2,3-triazole-4-carbonyl]-N-(3,4-difluorophenyl)piperidin-3-amine
3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
1-cyclopentyl-4-oxo-5-(4-phenylazepane-1-carbonyl)-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
8-(3-methylbutyl)-9-oxo-N-(thiophen-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxamide
(3S,4S)-4-(morpholin-4-yl)-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidin-3-ol
(3aS,6aS)-2-(cyclopropylmethyl)-5-(furan-2-ylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}thiophen-2-yl)ethan-1-one
2-{5-cyclopropyl-4-[4-(4-methylphenyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(5-methylfuran-2-yl)pyrimidine
(1S,4S)-2-(2-fluorophenyl)-5-[(2-hydroxynaphthalen-1-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
3-(3-chlorobenzoyl)-N-(2-methoxyphenyl)piperidine-1-carboxamide
1'-(3,4-dimethylbenzoyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-4-oxo-3,4-dihydroquinazoline-7-carboxamide
2-benzyl-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]-1,3-thiazole-4-carboxamide
5-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-methyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
2-(4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
5-ethyl-1'-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(4-fluorophenyl)-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-amine
1-[(1R,5R)-6-[(2,4-dimethoxy-3-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-ethyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(4-fluorophenyl)-N-{[1-(methoxymethyl)cyclopentyl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]-1-methyl-1H-pyrazole-5-carboxamide
N-[3-(dimethylamino)propyl]-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-methyl-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]-N-(2-methylphenyl)acetamide