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1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(pyridin-2-ylsulfanyl)propan-1-one
4-[(2R)-2-amino-2-phenylacetyl]-1-(4-methoxyphenyl)piperazin-2-one
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N-(2,3-dihydro-1H-inden-2-yl)-6,6-dimethyl-5-oxo-N-propylthiomorpholine-3-carboxamide
6-{1-[(2E)-3-(furan-2-yl)-2-phenylprop-2-enoyl]piperidin-3-yl}-2-methyl-3,4-dihydropyrimidin-4-one
3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
2-[1-(3-methylbutyl)-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperazin-2-yl]ethan-1-ol
ethyl 1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
4,6-dimethyl-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-2-oxo-1,2-dihydropyridine-3-carboxamide
3-butyl-1-methyl-4-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]piperazin-2-one
3-(2-methylpropyl)-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-5-carboxamide
N-(3,5-difluorophenyl)-3-hydroxy-3-(hydroxymethyl)pyrrolidine-1-carboxamide
2-(phenylsulfanyl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
3-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
3-[4-({[2-(2-chlorophenyl)ethyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
2-methoxy-4-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
2-[3-fluoro-5-(propan-2-yloxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-tert-butyl-4-[3-(3-methylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
N-(furan-2-ylmethyl)-3-({4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine-1-carboxamide
N-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)pyrrolidin-3-yl]methyl}propane-1-sulfonamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
4-(4-{[(5-fluoro-1H-indol-2-yl)methyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
3-chloro-4-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
4-cyclopentyl-N-[3-(dimethylamino)propyl]pyrimidin-2-amine
6-hydroxy-N-(2-methyl-1-benzofuran-5-yl)-1,4-oxazepane-4-carboxamide
(3S,4S)-4-(morpholin-4-yl)-1-[(trimethylpyrazin-2-yl)methyl]pyrrolidin-3-ol
N,N-bis(1,3-oxazol-4-ylmethyl)-3-(pyridin-4-yl)propanamide
6-chloro-4-(1,4-oxazepane-4-carbonyl)-2-(1H-pyrazol-4-yl)quinoline
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-(pyridin-3-yl)propanamide
N-cyclopropyl-3-(3-methoxyphenyl)-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrazole-4-carboxamide
ethyl 3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,3-dichlorophenyl)urea
N-[2-(dimethylamino)ethyl]-3-hydroxy-N-[(3-methylthiophen-2-yl)methyl]pyridine-2-carboxamide
2-{2-[2-(2,3-difluorophenyl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
(4aR,8aR)-2-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
1-({2-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]phenyl}methyl)piperidine-4-carboxamide
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-1-cyclopropyl-6-oxopiperidine-3-carboxamide
methyl (2S)-2-{[5-(2,5-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}-3-methylbutanoate
N-{2-[5-(4-acetylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
N,N-dimethyl-2-[(1S,5R)-6-(4-oxo-3,4-dihydroquinazoline-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N-[5-(morpholin-4-yl)pentyl]-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-{[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-6-azaspiro[2.5]octane
3-[methyl({2-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl})amino]-1λ6-thiolane-1,1-dione
5-{1-[(3E)-pent-3-enoyl]pyrrolidin-2-yl}-N-[2-(pyrazin-2-yl)ethyl]thiophene-2-carboxamide
ethyl 4-{1-[(5-chloro-2,3-dimethoxyphenyl)methyl]piperidin-3-yl}piperazine-1-carboxylate
methyl 3-{4-cyclohexanecarbonyl-6-[(3-methoxyphenyl)methoxy]-2-oxo-1,4-diazepan-1-yl}propanoate
(1-{2-[2-(isoquinolin-5-yl)-1H-imidazol-1-yl]ethyl}piperidin-2-yl)methanol
N,N-dimethyl-4-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)benzamide
({4-[4-(4-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-1,3-thiazol-2-yl}methyl)dimethylamine