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2-(dimethylamino)-2-(4-methylphenyl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]acetamide
4-(furan-2-carbonyl)-2-(2-phenylethyl)morpholine
N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
6-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane-6-carbonyl}-2,3,4,9-tetrahydro-1H-carbazole
1-methyl-3-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1,2,5,6,7,8-hexahydroquinolin-2-one
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-methoxypiperidine
8-[(dimethyl-1,3-thiazol-5-yl)methyl]-8-azaspiro[4.5]decane-7,9-dione
4-methyl-6-(4-{[1-(thiophen-3-yl)propan-2-yl]amino}piperidin-1-yl)pyrimidin-2-amine
N-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}methyl)methanesulfonamide
4-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2,6-dimethylpyridine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}piperidin-2-one
dimethyl({2-[(6-phenylpyridazin-3-yl)oxy]phenyl}methyl)amine
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-N'-(2-fluoro-5-methylphenyl)butanediamide
[(1-benzyl-1H-imidazol-2-yl)methyl]({[2-(furan-2-yl)pyrimidin-5-yl]methyl})methylamine
[1-(2-methanesulfonylethyl)-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
(2S,4R)-4-(dimethylamino)-1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrrolidine-2-carboxylic acid
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
4-benzyl-3-ethyl-1-(2-methoxyacetyl)-1,4-diazepan-5-one
N-cyclopropyl-5-methyl-4-{[(6-methylpyridin-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
[3-(3-phenylpropyl)-1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-3-yl]methanol
3-[(3R,4S)-1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
(1R,5S,8S)-8-methoxy-N-[4-(1H-pyrazol-1-yl)phenyl]-3-azabicyclo[3.2.1]octane-3-carboxamide
8-(1-aminocyclopropanecarbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[(2-fluorophenyl)formamido]-N-methyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]propanamide
6-[2-(4-fluorophenyl)piperidine-1-carbonyl]-1H-indole
1-ethyl-3-(3-fluoro-5-methylphenyl)-1-[2-(4-methylbenzenesulfonyl)ethyl]urea
2-(4-fluorophenoxy)-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-(1H-pyrazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-4-[(2-hydroxyethyl)(methyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid
N-methyl-N-(propan-2-yl)-2-(pyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N,2,4-trimethyl-1,3-thiazole-5-carboxamide
4-[5-(2-chloro-6-methylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]morpholine
N2-[3-(4-methoxyphenoxy)propyl]-N2-methylpyrrolidine-1,2-dicarboxamide
4-{[3-(4-fluorophenoxymethyl)piperidin-1-yl]methyl}-2-methoxyphenol
1-(3-cyano-4-methoxyphenyl)-3-[3-(oxolan-3-yl)propyl]urea
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[2-(morpholin-4-yl)ethyl]propanamide
2-[3-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)phenyl]ethan-1-amine
methyl (3S)-3-amino-4-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-oxobutanoate
4-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperazin-1-yl)benzoic acid
N-(1-methyl-1H-pyrazol-4-yl)-2-[3-(2-phenylacetyl)piperidin-1-yl]acetamide
2-amino-1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
(2S,4S)-1-benzyl-N-ethyl-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
1-(4-{4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazin-1-yl}piperidin-1-yl)butan-1-one
5-methyl-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-3-phenyl-1,2-oxazole-4-carboxamide
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}[3-(2-methyl-1H-imidazol-1-yl)propyl]amine
1-(4-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
1-(cyclobutylmethyl)-4-[(2,3-dimethoxyphenyl)methyl]piperazine
1-(4-chlorophenyl)-N-(1H-imidazol-2-ylmethyl)cyclobutane-1-carboxamide