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1-(cyclopropylmethyl)-4-(5-methylpyridine-3-carbonyl)-2-(propan-2-yl)-1,4-diazepane
1-methanesulfonyl-4-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-1,4-diazepane
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]ethan-1-one
(3aS,6aR)-5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-{[(3,5-dimethoxyphenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-3-(pyridin-4-yl)propan-1-one
3-(pyrrolidin-1-yl)-1-{[4-(trifluoromethyl)phenyl]methyl}piperidine
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(pyridin-4-ylmethyl)acetamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(3-methylbutyl)amino]methyl}piperidin-2-one
(3S,4S)-4-(morpholin-4-yl)-1-[2-(phenylamino)pyrimidine-5-carbonyl]pyrrolidin-3-ol
1-{5-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
(2S,4S)-4-amino-1-(3-methylbut-2-enoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
6-[6-hydroxy-4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]pyrazine-2-carboxamide
2-{2-[2-(4-fluorophenyl)pyrrolidin-1-yl]ethoxy}ethan-1-ol
[(3R,4R)-1-(4-ethylbenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
4-(2-methyl-1H-imidazol-1-yl)-1-{[(2-methylphenyl)methyl]carbamoyl}piperidine-4-carboxylic acid
1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-pyrazol-1-yl)propan-1-one
4-(2,5-dimethoxybenzoyl)-N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
(2S)-2-cyclohexyl-2-{[3-(2-fluorophenyl)-1H-pyrazol-5-yl]formamido}acetic acid
ethyl 1-[(2H-1,3-benzodioxol-5-yl)carbamoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
methyl 4-oxo-4-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}butanoate
5-(2-methylpropyl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-3-carboxamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
2-[2-(furan-3-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-6-methylpyridine
(1S,5R)-6-(cyclopropylmethyl)-3-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-ethyl-6-methyl-2-oxo-N-[(2-phenoxypyridin-3-yl)methyl]-1,2-dihydropyridine-3-carboxamide
1-[(4aR,8aR)-4a-hydroxy-7-{[4-(3-methylphenyl)phenyl]methyl}-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
2-(1-{[1-(quinolin-5-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
5-ethyl-N,2-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-4-amine
8-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(2,2,3,3-tetrafluoropropoxy)acetamide
2-methoxy-1-(1'-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
8-[3-(furan-2-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(2-{1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]piperidin-2-yl}ethyl)morpholine
4-[4-(benzyloxy)butyl]-1,2-dihydropyridin-2-one
6-[4-(1-ethoxyethyl)phenyl]-N,N-dimethylpyridine-3-carboxamide
(2E)-N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-3-(3-fluorophenyl)-N-(pyridin-3-ylmethyl)prop-2-enamide
methyl 3-{[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]amino}benzoate
4-(1H-imidazol-2-yl)-1-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-1,2,3-triazole
methyl(pyridin-3-ylmethyl)[2-(quinoxalin-2-yloxy)hex-5-en-1-yl]amine
2-(4-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenoxy)ethan-1-ol
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
4-(4-benzyl-1H-1,2,3-triazol-1-yl)-1-(thian-4-yl)piperidine
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methoxypiperidine
2-methyl-7-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-(3,4-dimethoxyphenyl)-1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-3-amine
4-({2-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-3-methyl-1-oxobutan-2-yl)acetamide